SCHEMBL5268084

SCHEMBL5268084

Cc1nc(N2CC(CNC(=O)NS(=O)(=O)c3ccc(Cl)s3)C2)c(C#N)cc1C(=O)O

nearest known ligand 0.66

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
P2RY12 Q9H244 18/20 0.66
CYP3A4 P08684 3/20 0.45
CYP2C9 P11712 3/20 0.45
CYP1A2 P05177 2/20 0.45
CYP2D6 P10635 2/20 0.45
CYP2C19 P33261 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4105134 0.91 P2RY12 (0.81) P2RY12CYP3A4CYP2C9
SCHEMBL5592539 0.89 P2RY12 (0.65) P2RY12CYP3A4CYP2C9CYP1A2CYP2D6
SCHEMBL29258649 0.86 P2RY12 (0.81) P2RY12CYP3A4CYP2C9CYP1A2CYP2D6
SCHEMBL5264696 0.85 P2RY12 (0.65) P2RY12CYP3A4CYP2C9
SCHEMBL29258458 0.82 P2RY12 (0.74) P2RY12CYP3A4CYP2C9CYP1A2CYP2D6
SCHEMBL4109942 0.81 P2RY12 (0.81) P2RY12CYP3A4CYP2C9CYP1A2CYP2D6
SCHEMBL4098259 0.80 P2RY12 (1.00) P2RY12CYP3A4CYP2C9
SCHEMBL4105892 0.80 P2RY12 (0.80) P2RY12CYP3A4CYP2C9
SCHEMBL5315088 0.78 P2RY12 (0.69) P2RY12CYP3A4CYP2C9CYP1A2CYP2D6
SCHEMBL5599353 0.78 P2RY12 (0.82) P2RY12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1836189-A1 NOVEL PYRIDINE COMPOUNDS AstraZeneca AB (SE) 2007-09-26 EP disclosed
WO-2006073361-A9 NOVEL PYRIDINE COMPOUNDS ASTRAZENECA AB (SE) 2007-08-02 WO disclosed
WO-2006073361-A1 NOVEL PYRIDINE COMPOUNDS ASTRAZENECA AB (SE) 2006-07-13 WO disclosed