SCHEMBL5265079

SCHEMBL5265079

O=C(O)c1cccnc1-c1nc(C(F)(F)F)ccc1C(=O)O

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.64
TDP1 Q9NUW8 2/20 0.64
TAS2R14 Q9NYV8 2/20 0.49
NAPRT Q6XQN6 2/20 0.47
TGFBR1 P36897 1/20 0.46
ALDH1A1 P00352 5/20 0.45
CYP3A4 P08684 2/20 0.45
MAPT P10636 1/20 0.45
ALOX15 P16050 1/20 0.45
TSHR P16473 1/20 0.45
BLM P54132 1/20 0.45
AGER Q15109 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
LMNA P02545 3/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
RUNX1 Q01196 1/20 0.44
DHODH Q02127 4/20 0.42
MEN1 O00255 1/20 0.42
GMNN O75496 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5265077 0.82 TAS2R14 (0.47) KDM4ETDP1TAS2R14TGFBR1BLM
SCHEMBL30639802 0.82 KDM4E (0.95) KDM4ETDP1NAPRTALDH1A1CYP3A4
SCHEMBL30639818 0.82 KDM4E (0.95) KDM4ETDP1NAPRTALDH1A1CYP3A4
Trifluoroacetic Acid SCHEMBL5691131 0.80 KDM4E (0.78) KDM4ETDP1NAPRTALDH1A1CYP3A4
SCHEMBL270419 0.80 KDM4E (1.00) KDM4ETDP1NAPRTALDH1A1CYP3A4
SCHEMBL13853227 0.80 TAS2R14 (0.48) KDM4ETAS2R14ALDH1A1LMNADHODH
SCHEMBL29723448 0.78 KDM4E (0.95) KDM4ETDP1NAPRTALDH1A1CYP3A4
SCHEMBL5263715 0.74 CYP1A2 (0.43) KDM4ETDP1TAS2R14TGFBR1ALDH1A1
SCHEMBL13853224 0.74 CSNK1D (0.41) KDM4ETAS2R14DHODHPTGS1PTGS2
SCHEMBL4197626 0.74 TDP1 (0.61) KDM4ETDP1NAPRTALDH1A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1824828-A2 PYRIDINE BASED COMPOUNDS USEFUL AS INTERMEDIATES FOR PHARMACEUTICAL OR AGRICULTURAL END-PRODUCTS Peakdale Molecular Limited (GB) 2007-08-29 EP claimed
WO-2006059103-A2 PYRIDINE BASED COMPOUNDS USEFUL AS INTERMEDIATES FOR PHARMACEUTICAL OR AGRICULTURAL END-PRODUCTS PEAKDALE MOLECULAR LIMITED (GB) 2006-06-08 WO claimed