SCHEMBL5265487

SCHEMBL5265487

COc1ccc(C(c2ccccn2)n2c(=O)ccc3cnc(Nc4ccc(N5CCCCC5)cc4)nc32)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 18/20 0.53
CCND1 P24385 18/20 0.53
CCND2 P30279 12/20 0.53
CCND3 P30281 12/20 0.53
CDK2 P24941 7/20 0.52
CCNA2 P20248 6/20 0.52
CCNE1 P24864 5/20 0.52
CCNE2 O96020 4/20 0.52
CCNA1 P78396 4/20 0.52
FGFR4 P22455 4/20 0.52
CCNB2 O95067 3/20 0.52
CDK1 P06493 3/20 0.52
CCNB1 P14635 3/20 0.52
CCNB3 Q8WWL7 3/20 0.52
FGFR1 P11362 3/20 0.52
FGFR2 P21802 3/20 0.52
FGFR3 P22607 3/20 0.52
EGFR P00533 1/20 0.46
KDR P35968 1/20 0.46
PAK4 O96013 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5265870 0.93 CDK4 (0.62) CDK4CCND1CCND2CCND3CDK2
SCHEMBL6808803 0.91 CDK4 (0.55) CDK4CCND1CCND2CCND3CDK2
SCHEMBL5267373 0.89 CDK4 (0.59) CDK4CCND1CCND2CCND3CDK2
SCHEMBL5266416 0.86 CDK4 (0.47) CDK4CCND1CCND2CCND3CDK2
SCHEMBL5263464 0.85 CDK4 (0.61) CDK4CCND1CCND2CCND3CDK2
SCHEMBL6807957 0.84 CDK4 (0.65) CDK4CCND1CCND2CCND3CDK2
SCHEMBL5263255 0.83 CDK4 (0.63) CDK4CCND1CCND2CCND3CDK2
SCHEMBL5266676 0.80 CDK4 (0.61) CDK4CCND1CCND2CCND3CDK2
SCHEMBL6802701 0.80 CDK4 (0.61) CDK4CCND1CCND2CCND3CDK2
SCHEMBL5263432 0.79 CDK4 (0.58) CDK4CCND1CCND2CCND3CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1806348-A2 Pyrido (2,3-D)Pyrimidines as inhibitors of cellular proliferation Warner-Lambert Company LLC (US) 2007-07-11 EP disclosed
US-6498163-B1 POTENT INHIBITORS OF CYCLIN-DEPENDENT KINASES AND GROWTH FACTOR MEDIATED KINASES; CANCER, RESTENOSIS, ATHEROSCLEROSIS WARNER-LAMBERT COMPANY 2002-12-24 US disclosed