SCHEMBL5267103

SCHEMBL5267103

COc1ccc2cccc(C(O)CN3CCCC(CNCC4=NC=CCC4)C3)c2n1

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 4/20 0.37
GHSR Q92847 1/20 0.35
SLC2A1 P11166 5/20 0.34
PRMT5 O14744 1/20 0.33
WDR77 Q9BQA1 1/20 0.33
HTT P42858 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.32
MTNR1A P48039 2/20 0.32
MTNR1B P49286 2/20 0.32
SLC6A2 P23975 1/20 0.31
SLC6A4 P31645 1/20 0.31
SLC6A3 Q01959 1/20 0.31
MCHR1 Q99705 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
KDM2B Q8NHM5 1/20 0.31
HTR2C P28335 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5265408 0.89 KCNH2 (0.40) KCNH2SLC2A1SLC6A2SLC6A4SLC6A3
SCHEMBL5315739 0.80 KCNH2 (0.45) KCNH2SLC2A1SMN1; SMN2
SCHEMBL5262236 0.79 KCNH2 (0.58) KCNH2SLC2A1
SCHEMBL5432954 0.75 KCNH2 (0.48) KCNH2
SCHEMBL5426370 0.75
SCHEMBL5264956 0.74 HTR1A (0.42) SLC6A4
SCHEMBL5317515 0.74 KCNH2 (0.34) KCNH2GHSRSLC2A1SMN1; SMN2MEN1
SCHEMBL5437147 0.74 SLC2A1 (0.32) KCNH2SLC2A1HTT
SCHEMBL7101571 0.71 KCNH2 (0.66) KCNH2SLC2A1
SCHEMBL4468563 0.70 KCNH2 (0.43) KCNH2SLC2A1PRMT5WDR77MTNR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1781650-A1 NOVEL COMPOUNDS HAVING AN ANTI-BACTERIAL ACTIVITY Morphochem Aktiengesellschaft Für Kombinatorische Chemie (DE) 2007-05-09 EP disclosed
WO-2006021448-A1 NOVEL COMPOUNDS HAVING AN ANTI-BACTERIAL ACTIVITY Morphochem Aktiengesellschaft für kombinatorische Chemie (DE) 2006-03-02 WO disclosed