SCHEMBL5267191

SCHEMBL5267191

CC(C)(C)Nc1c(-c2ccc(C#Cc3ccc(F)c(C#N)c3)s2)nc2ccccn12

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA1B P35368 1/20 0.44
TRPA1 O75762 3/20 0.41
BACE1 P56817 5/20 0.40
BACE2 Q9Y5Z0 5/20 0.40
TOP2A P11388 1/20 0.39
TRIM24 O15164 1/20 0.39
SALL4 Q9UJQ4 1/20 0.39
TRIM33 Q9UPN9 1/20 0.39
HDAC7 Q8WUI4 2/20 0.38
HDAC9 Q9UKV0 2/20 0.38
HDAC5 Q9UQL6 2/20 0.38
HDAC4 P56524 1/20 0.38
HDAC3 O15379 1/20 0.38
NCOR2 Q9Y618 1/20 0.38
MAPT P10636 3/20 0.38
GAA P10253 3/20 0.38
PKM P14618 2/20 0.38
TP53 P04637 1/20 0.38
PKLR P30613 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5128464 0.99 ADRA1B (0.44) ADRA1BTRPA1BACE1BACE2TOP2A
SCHEMBL5129775 0.90 ADRA1B (0.48) ADRA1BTRPA1BACE1BACE2TOP2A
SCHEMBL5266905 0.89 ADRA1B (0.47) ADRA1BTRPA1BACE1BACE2TOP2A
Hydrochloric Acid SCHEMBL5113165 0.88 ADRA1B (0.46) ADRA1BTRPA1BACE1BACE2TOP2A
SCHEMBL5117968 0.87 ADRA1B (0.48) ADRA1BTRPA1BACE1BACE2TOP2A
SCHEMBL5127195 0.85 ADRA1B (0.50) ADRA1BTRPA1BACE1BACE2TOP2A
SCHEMBL5117557 0.83 ADRA1B (0.48) ADRA1BTRPA1BACE1BACE2TOP2A
SCHEMBL5121270 0.82 ADRA1B (0.46) ADRA1BTRPA1BACE1BACE2TOP2A
Hydrochloric Acid SCHEMBL5121423 0.82 ADRA1B (0.45) ADRA1BTRPA1BACE1BACE2TOP2A
SCHEMBL5125295 0.81 BRD4 (0.42) TRPA1TRIM24SALL4TRIM33HDAC5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1791840-A1 SUBSTITUTED BICYCLIC IMIDAZO-3-YLAMINE COMPOUNDS Grünenthal GmbH (DE) 2007-06-06 EP claimed
WO-2006029980-A1 SUBSTITUTED BICYCLIC IMIDAZO-3-YLAMINE COMPOUNDS Grünenthal GmbH (DE) 2006-03-23 WO claimed
EP-1791840-A1 SUBSTITUTED BICYCLIC IMIDAZO-3-YLAMINE COMPOUNDS Grünenthal GmbH (DE) 2007-06-06 EP disclosed
WO-2006029980-A1 SUBSTITUTED BICYCLIC IMIDAZO-3-YLAMINE COMPOUNDS Grünenthal GmbH (DE) 2006-03-23 WO disclosed