SCHEMBL5267455

SCHEMBL5267455

O=C(COc1ccccc1)Nc1c[nH]nc1C(=O)NCc1ccco1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.63
TP53 P04637 2/20 0.63
HSD17B10 Q99714 4/20 0.59
TSHR P16473 2/20 0.59
KDM4E B2RXH2 1/20 0.59
ALDH1A1 P00352 9/20 0.52
HPGD P15428 6/20 0.52
MEN1 O00255 2/20 0.52
KMT2A Q03164 2/20 0.52
POLB P06746 5/20 0.52
MAPT P10636 5/20 0.50
L3MBTL1 Q9Y468 3/20 0.50
TDP1 Q9NUW8 2/20 0.50
ESR1 P03372 1/20 0.50
APEX1 P27695 1/20 0.50
LMNA P02545 1/20 0.50
MAPK1 P28482 2/20 0.49
USP2 O75604 1/20 0.48
ALOX15 P16050 1/20 0.48
HIF1A Q16665 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5269122 0.85 ALDH1A1 (0.54) SMN1; SMN2TP53HSD17B10TSHRALDH1A1
SCHEMBL5270571 0.85 KMT2A (0.59) SMN1; SMN2HSD17B10TSHRALDH1A1HPGD
SCHEMBL5265275 0.84 ALDH1A1 (0.54) SMN1; SMN2TP53HSD17B10TSHRKDM4E
SCHEMBL5270376 0.84 TSHR (0.50) SMN1; SMN2TP53HSD17B10TSHRKDM4E
SCHEMBL5270730 0.84 HPGD (0.69) SMN1; SMN2TP53HSD17B10TSHRKDM4E
SCHEMBL5266740 0.82 TDP1 (0.49) SMN1; SMN2TP53HSD17B10TSHRKDM4E
SCHEMBL4284612 0.82 ALDH1A1 (0.51) SMN1; SMN2TP53HSD17B10TSHRKDM4E
SCHEMBL5267614 0.81 ALDH1A1 (0.53) SMN1; SMN2TP53HSD17B10TSHRALDH1A1
SCHEMBL5269978 0.81 ALDH1A1 (0.54) SMN1; SMN2TP53TSHRKDM4EALDH1A1
SCHEMBL5268206 0.80 HPGD (0.53) TP53HSD17B10TSHRKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1847531-A1 PYRAZOLE COMPOUND Takeda Pharmaceutical Company Limited (JP) 2007-10-24 EP disclosed