SCHEMBL5274265

SCHEMBL5274265

O=C(C1=NN(c2ccc(Cl)cc2Cl)C(c2ccc(I)cc2)C1)N1CCCCCC1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 12/20 0.56
CNR2 P34972 9/20 0.56
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
CASP3 P42574 1/20 0.40
SENP8 Q96LD8 1/20 0.40
SENP7 Q9BQF6 1/20 0.40
SENP6 Q9GZR1 1/20 0.40
ALPL P05186 3/20 0.40
LMNA P02545 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
MAPT P10636 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
GPR55 Q9Y2T6 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4607380 0.95 CNR1 (0.61) CNR1CNR2NPC1RAB9ACASP3
SCHEMBL2018135 0.95 CNR1 (0.61) CNR1CNR2NPC1RAB9ACASP3
SCHEMBL2288238 0.95 CNR1 (0.61) CNR1CNR2NPC1RAB9ACASP3
SCHEMBL5275640 0.92 CNR2 (0.56) CNR1CNR2NPC1RAB9ACASP3
SCHEMBL8463209 0.92 CNR2 (0.50) CNR1CNR2CYP3A4CYP2D6CYP2C19
SCHEMBL2015954 0.91 CNR2 (0.62) CNR1CNR2NPC1RAB9ACASP3
SCHEMBL5273863 0.91 CNR1 (0.55) CNR1CNR2NPC1RAB9ACASP3
SCHEMBL5275927 0.91 CNR1 (0.55) CNR1CNR2NPC1RAB9ACASP3
SCHEMBL8472367 0.90 CNR1 (0.50) CNR1CNR2
SCHEMBL8453029 0.89 CNR2 (0.52) CNR1CNR2NPC1RAB9ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1849776-A1 Azepane- or Azocane-substituted pyrazoline compounds, their preparation and use as medicaments LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2007-10-31 EP disclosed