SCHEMBL8453029

SCHEMBL8453029

S=C(C1=NN(c2ccc(Cl)cc2Cl)C(c2ccc(I)cc2)C1)N1CCCCCCC1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 10/20 0.52
CNR1 P21554 10/20 0.52
LMNA P02545 3/20 0.39
NPC1 O15118 3/20 0.39
RAB9A P51151 3/20 0.39
MAPT P10636 3/20 0.39
HPGD P15428 3/20 0.39
ALDH1A1 P00352 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
TDP1 Q9NUW8 1/20 0.39
PKM P14618 1/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
PHGDH O43175 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4605553 0.94 CNR2 (0.58) CNR2CNR1LMNANPC1RAB9A
SCHEMBL4605163 0.94 CNR2 (0.58) CNR2CNR1LMNANPC1RAB9A
SCHEMBL5274265 0.89 CNR1 (0.56) CNR2CNR1LMNANPC1RAB9A
SCHEMBL4605679 0.87 CNR1 (0.60) CNR2CNR1LMNAMAPTCYP1A2
SCHEMBL4606201 0.87 CNR1 (0.60) CNR2CNR1LMNAMAPTCYP1A2
SCHEMBL4606979 0.86 CNR1 (0.53) CNR2CNR1
SCHEMBL8469991 0.86 CNR2 (0.49) CNR2CNR1
SCHEMBL4605885 0.85 CNR1 (0.61) CNR2CNR1LMNAMAPTCYP1A2
SCHEMBL4607380 0.83 CNR1 (0.61) CNR2CNR1NPC1RAB9AHPGD
SCHEMBL2288238 0.83 CNR1 (0.61) CNR2CNR1NPC1RAB9AHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1946777-A1 Substituted pyrazoline for preventing weight gain Laboratorios del Dr. Esteve S.A. (ES) 2008-07-23 EP disclosed