SCHEMBL527773

SCHEMBL527773

Cc1cc(NS(C)(=O)=O)ccc1-c1cc(OC(C)C)ccn1

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 11/20 0.47
EPHX2 P34913 1/20 0.41
NR1H4 Q96RI1 1/20 0.41
IKBKB O14920 1/20 0.40
CHUK O15111 1/20 0.40
KDM4E B2RXH2 1/20 0.39
SLC6A3 Q01959 2/20 0.37
SCN9A Q15858 1/20 0.37
FFAR4 Q5NUL3 1/20 0.36
PIK3CD O00329 1/20 0.36
PIK3CA P42336 1/20 0.36
PIK3CB P42338 1/20 0.36
PIK3CG P48736 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3375902 0.79 ACACB (0.49) CYP17A1EPHX2NR1H4IKBKBCHUK
SCHEMBL527462 0.74 CYP17A1 (0.66) CYP17A1SLC6A3
Lithium SCHEMBL31041157 0.71 CYP17A1 (0.63) CYP17A1KDM4E
SCHEMBL526763 0.70 CYP17A1 (0.53) CYP17A1KDM4E
SCHEMBL13950331 0.66 KMO (0.46) FFAR4
SCHEMBL526391 0.66 CYP17A1 (0.78) CYP17A1SLC6A3
SCHEMBL526999 0.66 CYP17A1 (0.72) CYP17A1
SCHEMBL4661111 0.65 CYP17A1 (0.56) CYP17A1IKBKBCHUKKDM4E
SCHEMBL11233535 0.64 PTGS1 (0.55) CYP17A1KDM4E
SCHEMBL527307 0.64 CYP17A1 (0.73) CYP17A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2598481-A1 SULFONAMIDE COMPOUNDS USEFUL AS CYP17 INHIBITORS Bristol-Myers Squibb Company (US) 2013-06-05 EP disclosed
WO-2012015723-A1 SULFONAMIDE COMPOUNDS USEFUL AS CYP17 INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2012-02-02 WO disclosed