SCHEMBL5285565

SCHEMBL5285565

O=S(=O)(O)C=Cc1nn(Cc2ccccc2)c2c1CS(=O)(=O)CC2

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 2/20 0.36
HDAC3 O15379 1/20 0.36
HDAC4 P56524 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC7 Q8WUI4 1/20 0.36
HDAC2 Q92769 1/20 0.36
HDAC10 Q969S8 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
HDAC9 Q9UKV0 1/20 0.36
HDAC5 Q9UQL6 1/20 0.36
KCNK3 O14649 3/20 0.35
HTR7 P34969 2/20 0.34
HTR1A P08908 1/20 0.34
HTR2A P28223 1/20 0.34
BRD4 O60885 1/20 0.33
EP300 Q09472 1/20 0.33
CREBBP Q92793 1/20 0.33
GAA P10253 1/20 0.33
TSHR P16473 1/20 0.33
MEN1 O00255 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3894535 1.00 HDAC6 (0.36) HDAC6HDAC3HDAC4HDAC1HDAC7
SCHEMBL4097112 0.83 MEN1 (0.43) KCNK3HTR7HTR1AHTR2ATSHR
SCHEMBL4097113 0.83 MEN1 (0.43) KCNK3HTR7HTR1AHTR2ATSHR
SCHEMBL13866959 0.82 CNR2 (0.41) HDAC6HDAC3HDAC4HDAC1HDAC7
SCHEMBL13866943 0.82 CNR2 (0.41) HDAC6HDAC3HDAC4HDAC1HDAC7
SCHEMBL4711770 0.82 HTR2C (0.34) HDAC6HDAC3HDAC4HDAC1HDAC7
SCHEMBL3889267 0.80 HDAC10 (0.35) HDAC6HDAC10KCNK3HTR7HTR1A
SCHEMBL3889272 0.80 HDAC10 (0.35) HDAC6HDAC10KCNK3HTR7HTR1A
SCHEMBL13866955 0.78 CNR2 (0.36) HDAC6HDAC3HDAC4HDAC1HDAC7
SCHEMBL13866952 0.78 CNR2 (0.36) HDAC6HDAC3HDAC4HDAC1HDAC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1863479-A1 TETRAHYDROTHIOPYRANO PYRAZOLE CANNABINOID MODULATORS CROSS REFERENCE TO RELATED APPLICATIONS JANSSEN PHARMACEUTICA N.V. (BE) 2007-12-12 EP disclosed
WO-2006107561-A1 TETRAHYDROTHIOPYRANO PYRAZOLE CANNABINOID MODULATORS JANSSEN PHARMACEUTICA, N.V. (BE) 2006-10-12 WO disclosed