SCHEMBL5285848

SCHEMBL5285848

COc1cccc(-c2cncc(O[C@H]3SC[C@@H](OC(C)=O)[C@H](OC(C)=O)[C@H]3OC(C)=O)c2)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 7/20 0.39
CYP11B2 P19099 7/20 0.39
KDR P35968 1/20 0.39
BRD4 O60885 1/20 0.37
CYP1A2 P05177 4/20 0.36
CYP3A4 P08684 3/20 0.36
CYP2C9 P11712 2/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
MKNK1 Q9BUB5 1/20 0.36
MKNK2 Q9HBH9 1/20 0.36
PIK3CG P48736 1/20 0.36
CYP2C19 P33261 1/20 0.35
ALDH1A1 P00352 1/20 0.35
HPGD P15428 1/20 0.35
ADORA3 P0DMS8 1/20 0.35
ADORA2B P29275 1/20 0.35
ADORA1 P30542 1/20 0.35
CHEK2 O96017 1/20 0.35
CTSA P10619 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2141882 1.00 CYP11B1 (0.39) CYP11B1CYP11B2KDRBRD4CYP1A2
SCHEMBL2412501 0.96 CYP11B1 (0.39) CYP11B1CYP11B2KDRBRD4CYP1A2
SCHEMBL2412498 0.96 CYP11B1 (0.39) CYP11B1CYP11B2KDRBRD4CYP1A2
SCHEMBL316434 0.92 MKNK1 (0.40) CYP11B1CYP11B2CYP1A2CYP3A4CYP2C9
SCHEMBL3399894 0.92 MKNK1 (0.40) CYP11B1CYP11B2CYP1A2CYP3A4CYP2C9
SCHEMBL2142952 0.90 MAP4K4 (0.42) CYP11B1CYP11B2CYP1A2CYP3A4CYP2C9
SCHEMBL2139085 0.90 CHRNB2 (0.36) CYP11B1CYP11B2KDRMKNK1MKNK2
SCHEMBL2139089 0.90 CHRNB2 (0.36) CYP11B1CYP11B2KDRMKNK1MKNK2
SCHEMBL2411954 0.88 S1PR1 (0.35) CYP11B1CYP11B2KDRBRD4PIK3CG
SCHEMBL2411957 0.88 S1PR1 (0.35) CYP11B1CYP11B2KDRBRD4PIK3CG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1861411-A2 NOVEL COMPOUNDS DERIVED FROM 5-THIOXYLOSE AND THERAPEUTIC USE THEREOF LABORATOIRES FOURNIER S.A. (FR) 2007-12-05 EP disclosed
WO-2006100413-A9 NOVEL COMPOUNDS DERIVED FROM 5-THIOXYLOSE AND THERAPEUTIC USE THEREOF FOURNIER LAB SA (FR) 2007-10-18 WO disclosed
WO-2006100413-A2 NOVEL COMPOUNDS DERIVED FROM 5-THIOXYLOSE AND THERAPEUTIC USE THEREOF LABORATOIRES FOURNIER S.A. (FR) 2006-09-28 WO disclosed