SCHEMBL5286047

SCHEMBL5286047

O=C1c2ccc(Nc3ccccc3CCO)cc2CCN1Cc1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 3/20 0.52
ACHE P22303 1/20 0.40
MAPK14 Q16539 6/20 0.39
ITGB3 P05106 2/20 0.39
ITGA2B P08514 2/20 0.39
DHPS P49366 1/20 0.38
HRH3 Q9Y5N1 1/20 0.38
MAPK13 O15264 1/20 0.37
MAPK12 P53778 1/20 0.37
MAPK11 Q15759 1/20 0.37
HDAC3 O15379 1/20 0.37
HDAC4 P56524 1/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC7 Q8WUI4 1/20 0.37
HDAC2 Q92769 1/20 0.37
HDAC10 Q969S8 1/20 0.37
HDAC11 Q96DB2 1/20 0.37
HDAC8 Q9BY41 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
HDAC9 Q9UKV0 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15712413 0.79 GRM5 (0.51) GRM5ACHEMAPK14ITGB3ITGA2B
SCHEMBL5284549 0.78 MAPK14 (0.58) GRM5MAPK14
SCHEMBL7535369 0.78 GRM5 (0.62) GRM5ACHEITGB3ITGA2BDHPS
SCHEMBL15712412 0.76 GRM5 (0.48) GRM5MAPK14ITGB3ITGA2BALDH1A1
SCHEMBL3054839 0.74 GRM5 (0.67) GRM5ACHEITGB3ITGA2BDHPS
SCHEMBL29438631 0.74 GRM5 (0.67) GRM5ACHEITGB3ITGA2BDHPS
SCHEMBL5285908 0.72 MAPK14 (0.41) MAPK14MAPK13MAPK12MAPK11
SCHEMBL5303157 0.72 HDAC1 (0.54) MAPK14MAPK13MAPK12MAPK11HDAC3
SCHEMBL5946784 0.71 GRM5 (0.67) GRM5ACHEDHPSHRH3ALDH1A1
SCHEMBL7533063 0.71 GRM5 (0.67) GRM5ACHEHRH3ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007000337-A1 BICYCLIC DERIVATIVES AS P38 KINASE INHIBITORS PALAU PHARMA, S.A. (ES) 2007-01-04 WO claimed
WO-2007000337-A1 BICYCLIC DERIVATIVES AS P38 KINASE INHIBITORS PALAU PHARMA, S.A. (ES) 2007-01-04 WO disclosed