SCHEMBL528895

SCHEMBL528895

[c]1ccc(Nc2ccnc3ccccc23)cc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERBB2 P04626 1/20 0.61
HTT P42858 1/20 0.60
FADS1 O60427 1/20 0.57
EGFR P00533 1/20 0.57
DNMT1 P26358 4/20 0.57
DNMT3A Q9Y6K1 3/20 0.57
HDAC3 O15379 1/20 0.57
ACHE P22303 1/20 0.57
HDAC1 Q13547 1/20 0.57
HDAC7 Q8WUI4 1/20 0.57
HDAC2 Q92769 1/20 0.57
HDAC8 Q9BY41 1/20 0.57
HDAC6 Q9UBN7 1/20 0.57
HDAC9 Q9UKV0 1/20 0.57
HDAC5 Q9UQL6 1/20 0.57
DNMT3L Q9UJW3 1/20 0.57
GAK O14976 1/20 0.54
RIPK2 O43353 1/20 0.54
COQ8A Q8NI60 1/20 0.54
NLK Q9UBE8 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30420824 0.86 ERBB2 (0.73) ERBB2HTTFADS1EGFRDNMT1
SCHEMBL170830 0.86 ERBB2 (0.73) ERBB2HTTFADS1EGFRDNMT1
SCHEMBL5306062 0.83 DNMT1 (0.68) ERBB2HTTFADS1EGFRDNMT1
SCHEMBL6752938 0.82 HTR1A (0.68) ERBB2HTTFADS1EGFRDNMT1
SCHEMBL12217976 0.80 HTT (0.68) ERBB2HTTFADS1EGFRDNMT1
SCHEMBL4813919 0.80 DNMT1 (0.73) ERBB2HTTFADS1EGFRDNMT1
SCHEMBL12240670 0.80 HTT (0.68) ERBB2HTTFADS1EGFRDNMT1
SCHEMBL31197381 0.80 ALK (0.72) ERBB2HTTFADS1EGFRDNMT1
SCHEMBL15923366 0.80 ALK (0.72) ERBB2HTTFADS1EGFRDNMT1
SCHEMBL15673390 0.80 ERBB2 (0.66) ERBB2HTTFADS1EGFRDNMT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2597955-A1 QUINOLINE DERIVATIVES AND MELK INHIBITORS CONTAINING THE SAME OncoTherapy Science, Inc. (JP) 2013-06-05 EP disclosed
WO-2012016082-A1 QUINOLINE DERIVATIVES AND MELK INHIBITORS CONTAINING THE SAME ONCOTHERAPY SCIENCE, INC. (JP) 2012-02-02 WO disclosed