SCHEMBL5290068

SCHEMBL5290068

CCC=C(c1nc2cc(-c3ncc[nH]3)ccc2[nH]1)c1nc2cc(-c3ncc[nH]3)ccc2[nH]1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP19A1 P11511 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
NISCH Q9Y2I1 2/20 0.38
TLR9 Q9NR96 1/20 0.38
TLR8 Q9NR97 1/20 0.38
TLR7 Q9NYK1 1/20 0.38
VCP P55072 9/20 0.37
PARP1 P09874 1/20 0.37
PDE4A P27815 2/20 0.36
PDE4B Q07343 2/20 0.36
PDE4C Q08493 2/20 0.36
PDE4D Q08499 2/20 0.36
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 2/20 0.36
MTOR P42345 1/20 0.34
ADK P55263 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5290113 0.92 CYP3A4 (0.39) CYP1A2CYP3A4CYP2D6CYP19A1CYP2C9
SCHEMBL3830636 0.82 NISCH (0.38) CYP1A2CYP3A4CYP2D6CYP19A1CYP2C9
SCHEMBL3836383 0.82 NISCH (0.36) CYP1A2CYP3A4CYP2D6CYP19A1CYP2C9
SCHEMBL4706526 0.81 ALK (0.35)
SCHEMBL549271 0.78 NISCH (0.34) CYP1A2CYP3A4CYP2D6CYP19A1CYP2C9
SCHEMBL549270 0.78 NISCH (0.34) CYP1A2CYP3A4CYP2D6CYP19A1CYP2C9
SCHEMBL5307575 0.75 NISCH (0.51) CYP1A2CYP3A4CYP2D6CYP19A1CYP2C9
SCHEMBL548311 0.75 CYP1A2 (0.39) CYP1A2CYP3A4CYP2D6CYP19A1CYP2C9
SCHEMBL548310 0.75 CYP1A2 (0.39) CYP1A2CYP3A4CYP2D6CYP19A1CYP2C9
SCHEMBL7834814 0.75 TDP1 (0.46) CYP1A2CYP3A4CYP2D6CYP19A1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1858860-A1 PHTHALAZINONES Merck Patent GmbH (DE) 2007-11-28 EP disclosed
WO-2006097176-A1 PHTHALAZINONES MERCK PATENT GMBH (DE) 2006-09-21 WO disclosed