SCHEMBL529303

SCHEMBL529303

CCOC(=O)c1cnc2ccc(Br)cc2c1N(C)C1CCNCC1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXFP1 Q9HBX9 3/20 0.52
GAA P10253 2/20 0.52
NPSR1 Q6W5P4 1/20 0.52
MAPK1 P28482 1/20 0.52
JAK3 P52333 2/20 0.49
MEN1 O00255 4/20 0.48
KMT2A Q03164 4/20 0.48
ATM Q13315 1/20 0.48
PDE4B Q07343 1/20 0.47
LMNA P02545 1/20 0.46
MAPT P10636 1/20 0.46
ALDH1A1 P00352 2/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
AURKB Q96GD4 2/20 0.45
AURKA O14965 1/20 0.45
JAK1 P23458 1/20 0.44
NMT2 O60551 1/20 0.43
NMT1 P30419 1/20 0.43
GABRA1 P14867 1/20 0.43
GABRB1 P18505 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15191075 0.91 RXFP1 (0.55) RXFP1GAANPSR1MAPK1JAK3
SCHEMBL529843 0.88 RXFP1 (0.52) RXFP1GAANPSR1MAPK1JAK3
SCHEMBL528737 0.83 RXFP1 (0.49) RXFP1GAANPSR1MAPK1JAK3
SCHEMBL531700 0.82 MAPK1 (0.62) RXFP1GAANPSR1MAPK1MEN1
SCHEMBL529799 0.80 MAPK1 (0.49) RXFP1GAANPSR1MAPK1JAK3
SCHEMBL15190721 0.80 MAPK1 (0.63) RXFP1GAANPSR1MAPK1JAK3
SCHEMBL15191195 0.78 MAPK1 (0.66) RXFP1GAANPSR1MAPK1MEN1
SCHEMBL10681872 0.75 MEN1 (0.55) RXFP1GAANPSR1MAPK1MEN1
SCHEMBL23634709 0.75 MAPK1 (0.71) RXFP1GAANPSR1MAPK1MEN1
SCHEMBL15191143 0.75 MAPK1 (0.64) RXFP1GAANPSR1MAPK1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2597955-A1 QUINOLINE DERIVATIVES AND MELK INHIBITORS CONTAINING THE SAME OncoTherapy Science, Inc. (JP) 2013-06-05 EP disclosed
WO-2012016082-A1 QUINOLINE DERIVATIVES AND MELK INHIBITORS CONTAINING THE SAME ONCOTHERAPY SCIENCE, INC. (JP) 2012-02-02 WO disclosed