SCHEMBL529709

SCHEMBL529709

CC(=O)Cc1cnc2ccc(Br)cc2c1Cl

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 4/20 0.46
TSHR P16473 1/20 0.46
MALT1 Q9UDY8 2/20 0.44
RXFP1 Q9HBX9 2/20 0.42
CYP1A2 P05177 2/20 0.42
CYP2C9 P11712 2/20 0.42
CYP2C19 P33261 2/20 0.42
CYP2D6 P10635 1/20 0.42
MAPK1 P28482 1/20 0.40
GAA P10253 2/20 0.38
NPSR1 Q6W5P4 1/20 0.38
TNF P01375 1/20 0.38
ALDH1A1 P00352 4/20 0.38
CHEK1 O14757 1/20 0.37
PIM1 P11309 1/20 0.37
AKT1 P31749 1/20 0.37
FLT3 P36888 1/20 0.37
PIM3 Q86V86 1/20 0.37
MCL1 Q07820 1/20 0.37
CYP3A4 P08684 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27916351 0.83 MAPK1 (0.48) HTTTSHRMALT1RXFP1CYP1A2
SCHEMBL27916309 0.79 CYP1A2 (0.44) HTTTSHRMALT1RXFP1CYP1A2
SCHEMBL529214 0.78 HTT (0.63) HTTTSHRMALT1RXFP1CYP1A2
SCHEMBL529322 0.78 CYP1A2 (0.48) HTTTSHRMALT1RXFP1CYP1A2
SCHEMBL529686 0.77 CYP1A2 (0.40) HTTTSHRMALT1RXFP1CYP1A2
SCHEMBL28806276 0.77 CYP1A2 (0.40) HTTTSHRMALT1RXFP1CYP1A2
SCHEMBL529372 0.77 RXFP1 (0.43) HTTTSHRMALT1RXFP1CYP1A2
SCHEMBL529341 0.76 CYP1A2 (0.46) HTTTSHRMALT1RXFP1CYP1A2
SCHEMBL10282056 0.75 HTT (0.49) HTTTSHRMALT1RXFP1CYP1A2
SCHEMBL528765 0.75 RXFP1 (0.42) HTTTSHRMALT1RXFP1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2597955-A1 QUINOLINE DERIVATIVES AND MELK INHIBITORS CONTAINING THE SAME OncoTherapy Science, Inc. (JP) 2013-06-05 EP disclosed
WO-2012016082-A1 QUINOLINE DERIVATIVES AND MELK INHIBITORS CONTAINING THE SAME ONCOTHERAPY SCIENCE, INC. (JP) 2012-02-02 WO disclosed