SCHEMBL529686

SCHEMBL529686

O=CCc1cnc2ccc(Br)cc2c1Cl

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.40
CYP2D6 P10635 2/20 0.40
CYP2C9 P11712 2/20 0.40
CYP2C19 P33261 2/20 0.40
RXFP1 Q9HBX9 1/20 0.40
CHEK1 O14757 1/20 0.39
PIM1 P11309 1/20 0.39
AKT1 P31749 1/20 0.39
FLT3 P36888 1/20 0.39
PIM3 Q86V86 1/20 0.39
MALT1 Q9UDY8 2/20 0.38
TNF P01375 1/20 0.37
HTT P42858 7/20 0.37
LMNA P02545 4/20 0.37
ALDH1A1 P00352 3/20 0.37
KDM4E B2RXH2 3/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
HPGD P15428 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2718834 0.85 PARP1 (0.41) CYP1A2CYP2D6HTTLMNAKDM4E
SCHEMBL529947 0.82 HTT (0.39) RXFP1CHEK1PIM1AKT1FLT3
SCHEMBL2718102 0.82 PARP1 (0.39) MALT1HTTLMNAALDH1A1SMN1; SMN2
SCHEMBL27916309 0.81 CYP1A2 (0.44) CYP1A2CYP2D6CYP2C9CYP2C19RXFP1
SCHEMBL28072239 0.80 MALT1 (0.38) CYP1A2CYP2D6CYP2C9CYP2C19RXFP1
SCHEMBL28806276 0.79 CYP1A2 (0.40) CYP1A2CYP2D6CYP2C9CYP2C19RXFP1
SCHEMBL16730927 0.78 CYP1A2 (0.44) CYP1A2CYP2D6CYP2C9CYP2C19RXFP1
SCHEMBL2718503 0.78 ERN1 (0.42) CYP1A2CYP2C9CYP2C19ALDH1A1KDM4E
SCHEMBL529322 0.78 CYP1A2 (0.48) CYP1A2CYP2D6CYP2C9CYP2C19RXFP1
SCHEMBL529709 0.77 HTT (0.46) CYP1A2CYP2D6CYP2C9CYP2C19RXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2597955-A1 QUINOLINE DERIVATIVES AND MELK INHIBITORS CONTAINING THE SAME OncoTherapy Science, Inc. (JP) 2013-06-05 EP disclosed
WO-2012016082-A1 QUINOLINE DERIVATIVES AND MELK INHIBITORS CONTAINING THE SAME ONCOTHERAPY SCIENCE, INC. (JP) 2012-02-02 WO disclosed