SCHEMBL529835

SCHEMBL529835

CCOC(=O)NS(=O)(=O)Cl

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GAA P10253 3/20 0.42
MGAM O43451 1/20 0.42
SI P14410 1/20 0.42
MGAM2 Q2M2H8 1/20 0.42
ATM Q13315 1/20 0.41
SMN1; SMN2 Q16637 4/20 0.41
ALDH1A1 P00352 5/20 0.40
LMNA P02545 4/20 0.39
HSD17B10 Q99714 2/20 0.39
ALOX15 P16050 1/20 0.37
SOAT1 P35610 1/20 0.37
HTT P42858 1/20 0.37
CYP1A2 P05177 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
RECQL P46063 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5138578 0.81 GAA (0.46) GAAMGAMSIMGAM2ATM
SCHEMBL5228548 0.79 EPHX1 (0.48) ATMALDH1A1
SCHEMBL5639931 0.79 GAA (0.46) GAAMGAMSIMGAM2ATM
SCHEMBL3836989 0.79 GAA (0.44) GAAMGAMSIMGAM2SMN1; SMN2
SCHEMBL9574919 0.79 GAA (0.44) GAAMGAMSIMGAM2ATM
SCHEMBL23928061 0.77 GAA (0.42) GAAMGAMSIMGAM2ATM
SCHEMBL530163 0.77 FNTA (0.46) GAAMGAMSIMGAM2SMN1; SMN2
SCHEMBL25961960 0.77 GAA (0.42) GAAMGAMSIMGAM2SMN1; SMN2
SCHEMBL530162 0.77 GAA (0.42) GAAMGAMSIMGAM2ATM
SCHEMBL21420125 0.77 ATM (0.39) GAAMGAMSIMGAM2ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11319305-B2 Pyrimidine sulfamide derivative and preparation method and medical application thereof Shijiazhuang Sagacity New Drug Development Co., Ltd. (CN) 2022-05-03 US disclosed
CN-107427527-B Bile acid derivatives as FXR/TGR5 agonists and methods of use thereof 英安塔制药有限公司 2021-01-26 CN disclosed
US-20200283425-A1 PYRIMIDINE SULFAMIDE DERIVATIVE AND PREPARATION METHOD AND MEDICAL APPLICATION THEREOF Wuxi Biocity Biopharmaceutics Co., Ltd. (CN) 2020-09-10 US disclosed
EP-2598556-B1 PROCESS FOR PRODUCING SILOXANE COPOLYMERS WITH URETHANE-SULPHONAMIDO LINKING GROUPS WACKER CHEMIE AG (DE) 2014-09-03 EP disclosed
US-8741979-B2 Process for producing siloxane copolymers with urethane-sulphonamido linking groups WACKER CHEMIE AG (DE) 2014-06-03 US disclosed
EP-2598556-A1 PROCESS FOR PRODUCING SILOXANE COPOLYMERS WITH URETHANE-SULPHONAMIDO LINKING GROUPS Wacker Chemie AG (DE) 2013-06-05 EP disclosed
US-20130123376-A1 PROCESS FOR PRODUCING SILOXANE COPOLYMERS WITH URETHANE-SULPHONAMIDO LINKING GROUPS WACKER CHEMIE AG (DE) 2013-05-16 US disclosed
WO-2012013558-A1 PROCESS FOR PRODUCING SILOXANE COPOLYMERS WITH URETHANE-SULPHONAMIDO LINKING GROUPS WACKER CHEMIE AG (DE) 2012-02-02 WO disclosed
EP-0614887-B1 Indole-sulfonamides as antitumor agents LILLY CO ELI (US) 1997-06-11 EP disclosed
US-5565494-A BENZENESULFONYLUREA DERIVATIVES ELI LILLY AND COMPANY (US) 1996-10-15 US disclosed
WO-1994020101-A1 ANTITUMOR COMPOSITIONS AND METHODS OF TREATMENT ELI LILLY AND COMPANY (US) 1994-09-15 WO disclosed
EP-0614887-A1 Indole-sulfonamides as antitumor agents ELI LILLY AND COMPANY (US) 1994-09-14 EP disclosed
EP-0602878-A1 Diarylsulfonylureas and their use as antitumor agents ELI LILLY AND COMPANY (US) 1994-06-22 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130123376-A1 PROCESS FOR PRODUCING SILOXANE COPOLYMERS WITH URETHANE-SULPHONAMIDO LINKING GROUPS STS, MPST, IDUA GAA 288/4885MGAM 175/4885SI 16/4885
US-11319305-B2 Pyrimidine sulfamide derivative and preparation method and medical application thereof TBXA2R, P2RY11, TPMT GAA 2188/4885MGAM 3101/4885SI 864/4885
US-20200283425-A1 PYRIMIDINE SULFAMIDE DERIVATIVE AND PREPARATION METHOD AND MEDICAL APPLICATION THEREOF TBXA2R, P2RY11, TPMT GAA 2188/4885MGAM 3101/4885SI 864/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.