SCHEMBL5309151

SCHEMBL5309151

O=C(Nc1ccc(F)cc1)c1ccc(N2CCCN(C(=O)c3ccccc3C(F)(F)F)C2=O)nc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCD O00767 4/20 0.45
KMT2A Q03164 2/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
TRPV1 Q8NER1 1/20 0.42
SMN1; SMN2 Q16637 2/20 0.40
MAPT P10636 2/20 0.40
STAT3 P40763 1/20 0.40
ALDH1A1 P00352 2/20 0.40
CXCR2 P25025 2/20 0.40
KDM4E B2RXH2 1/20 0.40
PKM P14618 1/20 0.40
P4HTM Q9NXG6 1/20 0.40
GAA P10253 1/20 0.40
MAPK1 P28482 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
KCNQ3 O43525 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5308836 0.92 SCD (0.52) SCDTRPV1SMN1; SMN2MAPTP4HTM
SCHEMBL5313442 0.87 KCNQ3 (0.42) SCDKMT2ACYP1A2CYP3A4CYP2D6
SCHEMBL5307536 0.87 SCD (0.49) SCD
SCHEMBL5307037 0.86 SCD (0.45) SCDKMT2ATRPV1ALDH1A1KDM4E
SCHEMBL5309833 0.84 SCD (0.53) SCD
SCHEMBL5314446 0.84 SCD (0.48) SCDKMT2A
SCHEMBL5306749 0.84 F10 (0.47) SCDSMN1; SMN2
SCHEMBL5309747 0.84 SCD (0.43) SCDKMT2ATRPV1MAPTALDH1A1
SCHEMBL5309153 0.84 CYP1A2 (0.43) SCDKMT2ACYP1A2CYP3A4CYP2D6
SCHEMBL5309660 0.83 SCD (0.56) SCDSMN1; SMN2MAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007046867-A2 PIPERIDINE DERIVATIVES AND THEIR USES AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2007-04-26 WO disclosed