SCHEMBL5309153

SCHEMBL5309153

O=C(Nc1ccc(F)cc1)c1ccc(N2C=CCN(C(=O)c3ccccc3C(F)(F)F)C2=O)nc1

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
KMT2A Q03164 1/20 0.43
SCD O00767 4/20 0.42
CXCR2 P25025 4/20 0.40
P4HTM Q9NXG6 1/20 0.39
TRPV1 Q8NER1 1/20 0.39
HDAC1 Q13547 1/20 0.39
CA12 O43570 1/20 0.39
CA9 Q16790 1/20 0.39
CXCR1 P25024 1/20 0.38
CRACR2A Q9BSW2 1/20 0.38
MAPT P10636 1/20 0.38
STAT3 P40763 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5308839 0.92 SCD (0.49) SCDP4HTMTRPV1HDAC1CA12
SCHEMBL5313445 0.87 KCNQ3 (0.43) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL5307539 0.87 SCD (0.47) SCD
SCHEMBL5307042 0.86 SCD (0.42) KMT2ASCDTRPV1
SCHEMBL5309835 0.84 SCD (0.51) SCD
SCHEMBL5314447 0.84 SCD (0.46) KMT2ASCD
SCHEMBL5306753 0.84 SMN1; SMN2 (0.43) KMT2ASCDSMN1; SMN2
SCHEMBL5309749 0.84 SCD (0.41) KMT2ASCDTRPV1MAPT
SCHEMBL5309151 0.84 SCD (0.45) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL5309652 0.83 SCD (0.54) SCDSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007046867-A2 PIPERIDINE DERIVATIVES AND THEIR USES AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2007-04-26 WO disclosed