SCHEMBL5310025

SCHEMBL5310025

O=C1c2ccccc2CN1c1ccnc(Br)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.58
RAB9A P51151 4/20 0.58
CYP11B2 P19099 3/20 0.56
PKM P14618 3/20 0.52
TP53 P04637 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
KMT2A Q03164 2/20 0.44
LMNA P02545 2/20 0.44
MEN1 O00255 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C19 P33261 1/20 0.44
PGR P06401 1/20 0.44
CYP3A4 P08684 1/20 0.44
GAA P10253 1/20 0.44
NFKB1 P19838 1/20 0.44
DRD1 P21728 1/20 0.44
HTT P42858 1/20 0.44
NFKB2 Q00653 1/20 0.44
RELA Q04206 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11255826 0.79 NPC1 (0.74) NPC1RAB9ACYP11B2PKMTP53
SCHEMBL13113228 0.78 CYP11B2 (0.61) NPC1RAB9ACYP11B2PKMTP53
SCHEMBL28031462 0.78 NPC1 (0.68) NPC1RAB9ACYP11B2PKMTP53
Bromide SCHEMBL5310024 0.77 NPC1 (0.72) NPC1RAB9ACYP11B2PKMTP53
SCHEMBL29610632 0.75 NPC1 (0.74) NPC1RAB9ACYP11B2PKMTP53
SCHEMBL4150687 0.75 NPC1 (0.74) NPC1RAB9ACYP11B2PKMTP53
SCHEMBL2596828 0.75 MEN1 (0.49) TP53SMN1; SMN2KMT2AMEN1HTT
SCHEMBL4188221 0.74 NPC1 (1.00) NPC1RAB9ACYP11B2PKMTP53
SCHEMBL29874794 0.74 NPC1 (1.00) NPC1RAB9ACYP11B2PKMTP53
SCHEMBL8144026 0.74 NPC1 (0.64) NPC1RAB9ACYP11B2PKMTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007039146-A1 4-CARBOXY PYRAZOLE DERIVATIVES AS ANTI-VIRAL AGENTS SMITHKLINE BEECHAM CORPORATION (US) 2007-04-12 WO disclosed