SCHEMBL531059

SCHEMBL531059

CCCCCCNC(=O)CCc1cnc2ccccc2c1

nearest known ligand 0.61

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.61
HDAC3 O15379 4/20 0.53
HDAC1 Q13547 4/20 0.53
HDAC4 P56524 3/20 0.53
HDAC7 Q8WUI4 3/20 0.53
HDAC2 Q92769 3/20 0.53
HDAC10 Q969S8 3/20 0.53
HDAC11 Q96DB2 3/20 0.53
HDAC8 Q9BY41 3/20 0.53
HDAC6 Q9UBN7 3/20 0.53
HDAC9 Q9UKV0 3/20 0.53
HDAC5 Q9UQL6 3/20 0.53
TRPV1 Q8NER1 5/20 0.52
TRPM5 Q9NZQ8 1/20 0.51
ENPP2 Q13822 1/20 0.48
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12505085 0.88 TRPV1 (0.53) HPGDHDAC3HDAC1HDAC4HDAC7
SCHEMBL17954341 0.87 TRPV1 (0.51) HPGDHDAC3HDAC1HDAC4HDAC7
SCHEMBL30444584 0.83 EPHX2 (0.61) HDAC3HDAC1HDAC4HDAC7HDAC2
SCHEMBL30445391 0.83 EPHX2 (0.61) HDAC3HDAC1HDAC4HDAC7HDAC2
SCHEMBL6115263 0.79 TRPV1 (0.58) TRPV1MEN1KMT2A
SCHEMBL6114751 0.79 TRPV1 (0.58) TRPV1MEN1KMT2A
SCHEMBL6114625 0.79 TRPV1 (0.58) TRPV1MEN1KMT2A
SCHEMBL6114969 0.79 TRPV1 (0.58) TRPV1MEN1KMT2A
SCHEMBL6114605 0.79 TRPV1 (0.58) TRPV1MEN1KMT2A
SCHEMBL6114660 0.79 TRPV1 (0.58) TRPV1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2597955-A1 QUINOLINE DERIVATIVES AND MELK INHIBITORS CONTAINING THE SAME OncoTherapy Science, Inc. (JP) 2013-06-05 EP disclosed
WO-2012016082-A1 QUINOLINE DERIVATIVES AND MELK INHIBITORS CONTAINING THE SAME ONCOTHERAPY SCIENCE, INC. (JP) 2012-02-02 WO disclosed