SCHEMBL5312809

SCHEMBL5312809

CC(C)(C)OC(=O)NC[C@H](Cn1ccnc1[N+](=O)[O-])ON

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.44
LMNA P02545 1/20 0.42
THRB P10828 1/20 0.42
CYP2C19 P33261 1/20 0.42
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
OPRK1 P41145 1/20 0.40
CA12 O43570 9/20 0.39
CA1 P00915 9/20 0.39
CA2 P00918 9/20 0.39
CA9 Q16790 9/20 0.39
PCSK9 Q8NBP7 1/20 0.36
SERPINE1 P05121 1/20 0.35
TYMP P19971 3/20 0.34
CCR10 P46092 2/20 0.32
MEN1 O00255 1/20 0.31
ALDH1A1 P00352 1/20 0.31
MAPT P10636 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3835875 1.00 KMT2A (0.44) KMT2ALMNATHRBCYP2C19CYP3A4
SCHEMBL3840446 0.86 KMT2A (0.55) KMT2ALMNATHRBCYP2C19CYP3A4
SCHEMBL5314986 0.86 KMT2A (0.55) KMT2ALMNATHRBCYP2C19CYP3A4
SCHEMBL3839361 0.82 CYP3A4 (0.41) KMT2ALMNATHRBCYP2C19CYP3A4
SCHEMBL5312527 0.82 CYP3A4 (0.41) KMT2ALMNATHRBCYP2C19CYP3A4
SCHEMBL5329483 0.81 CA12 (0.40) KMT2ALMNATHRBCYP2C19CYP3A4
SCHEMBL31420756 0.79 CA12 (0.52) KMT2ALMNATHRBCYP2C19CYP3A4
SCHEMBL5315278 0.78 KMT2A (0.35) KMT2ALMNATHRBCYP2C19CYP3A4
SCHEMBL19027341 0.77 LMNA (0.49) KMT2ALMNATHRBCYP2C19CYP3A4
SCHEMBL5310209 0.76 KMT2A (0.50) KMT2ALMNATHRBCYP2C19CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0629617-B2 Heteroatom-bearing ligands and metal complexes thereof BRACCO INT BV (NL) 2007-09-26 EP disclosed
EP-0629617-B1 Heteroatom-bearing ligands and metal complexes thereof BRACCO INT BV (NL) 1998-04-29 EP disclosed
US-5665329-A Heteroatom-bearing ligands and metal complexes thereof BRACCO INTERNATIONAL B.V. 1997-09-09 US disclosed
US-5656254-A Polyaza heteroatom-bearing ligands and metal complexes thereof for imaging or radiotherapy BRACCO INTERNATIONAL B.V. 1997-08-12 US disclosed
US-5627286-A Heteroatom-bearing ligands and metal complexes thereof BRACCO INTERNATIONAL B.V. 1997-05-06 US disclosed
US-5608110-A Heteroatom-bearing ligands and metal complexes thereof BRACCO INTERNATIONAL B.V. 1997-03-04 US disclosed
EP-0629617-A1 Heteroatom-bearing ligands and metal complexes thereof BRACCO International B.V. (NL) 1994-12-21 EP disclosed