SCHEMBL5313145

SCHEMBL5313145

CC(C)CSc1cccc(N)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 4/20 0.50
BACE1 P56817 1/20 0.49
MAOB P27338 2/20 0.46
CYP3A4 P08684 3/20 0.41
CASP1 P29466 2/20 0.41
RECQL P46063 1/20 0.41
CRBN Q96SW2 1/20 0.39
MTNR1A P48039 3/20 0.37
MTNR1B P49286 3/20 0.37
ALDH1A1 P00352 5/20 0.37
GAA P10253 1/20 0.37
TP53 P04637 1/20 0.36
KDM4E B2RXH2 1/20 0.36
MEN1 O00255 1/20 0.36
MAPT P10636 1/20 0.36
ALOX15 P16050 1/20 0.36
CASP7 P55210 1/20 0.36
KMT2A Q03164 1/20 0.36
CTSK P43235 1/20 0.35
MAP1LC3B Q9GZQ8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28032991 0.79 BACE1 (0.42) MAOABACE1MAOBCYP3A4CASP1
SCHEMBL18739045 0.78 MAOA (0.47) MAOAMAOBMTNR1AMTNR1BALDH1A1
SCHEMBL926391 0.78 CYP3A4 (0.46) MAOABACE1MAOBCYP3A4CASP1
SCHEMBL30426786 0.78 CYP3A4 (0.46) MAOABACE1MAOBCYP3A4CASP1
SCHEMBL22468935 0.78 BACE1 (0.44) MAOABACE1MAOBCYP3A4CASP1
SCHEMBL12394796 0.77 MAOA (0.46) MAOAMAOBCYP3A4MTNR1AMTNR1B
Hydrochloric Acid SCHEMBL2651523 0.76 CYP3A4 (0.44) MAOABACE1MAOBCYP3A4CASP1
SCHEMBL8260518 0.75 MAOA (0.48) MAOAMAOBCYP3A4MTNR1AMTNR1B
SCHEMBL21313338 0.75 CYP3A4 (0.48) MAOABACE1MAOBCYP3A4CASP1
Fluoride SCHEMBL1336700 0.74 MAOA (0.68) MAOAMAOBMTNR1AMTNR1BALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007064869-A2 CATALYSTS FOR ARYL SULFIDE SYNTHESIS AND METHOD OF PRODUCING ARYL SULFIDES YALE UNIVERSITY (US) 2007-06-07 WO disclosed
WO-2006102760-A1 INHIBITORS OF HISTONE DEACETYLASE METHYLGENE INC. (CA) 2006-10-05 WO disclosed