SCHEMBL5313338

SCHEMBL5313338

CC(C)(NOCCN)C(Cn1ccnc1[N+](=O)[O-])=NO

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.42
THRB P10828 1/20 0.42
CYP2C19 P33261 1/20 0.42
CA12 O43570 5/20 0.40
CA1 P00915 5/20 0.40
CA2 P00918 5/20 0.40
CA9 Q16790 5/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
OPRK1 P41145 1/20 0.40
KMT2A Q03164 2/20 0.37
TYMP P19971 3/20 0.33
NOS1 P29475 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5310671 0.90 CA12 (0.42) LMNATHRBCYP2C19CA12CA1
SCHEMBL5316178 0.85 LMNA (0.41) LMNATHRBCYP2C19CA12CA1
SCHEMBL5316184 0.85 LMNA (0.41) LMNATHRBCYP2C19CA12CA1
SCHEMBL5310701 0.83 LMNA (0.41) LMNATHRBCYP2C19CA12CA1
SCHEMBL5310693 0.83 LMNA (0.41) LMNATHRBCYP2C19CA12CA1
SCHEMBL8365952 0.80 LMNA (0.48) LMNATHRBCYP2C19CA12CA1
SCHEMBL8365954 0.80 LMNA (0.48) LMNATHRBCYP2C19CA12CA1
SCHEMBL8764264 0.79 LMNA (0.49) LMNATHRBCYP2C19CA12CA1
SCHEMBL5315494 0.79 CA12 (0.41) LMNATHRBCYP2C19CA12CA1
SCHEMBL5312473 0.76 LMNA (0.48) LMNATHRBCYP2C19CA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0629617-B2 Heteroatom-bearing ligands and metal complexes thereof BRACCO INT BV (NL) 2007-09-26 EP disclosed
EP-0629617-B1 Heteroatom-bearing ligands and metal complexes thereof BRACCO INT BV (NL) 1998-04-29 EP disclosed
US-5741912-A DIAGNOSIS, THERAPY BRACCO INTERNATIONAL B.V. 1998-04-21 US disclosed
US-5665329-A Heteroatom-bearing ligands and metal complexes thereof BRACCO INTERNATIONAL B.V. 1997-09-09 US disclosed
US-5656254-A Polyaza heteroatom-bearing ligands and metal complexes thereof for imaging or radiotherapy BRACCO INTERNATIONAL B.V. 1997-08-12 US disclosed
US-5627286-A Heteroatom-bearing ligands and metal complexes thereof BRACCO INTERNATIONAL B.V. 1997-05-06 US disclosed
US-5608110-A Heteroatom-bearing ligands and metal complexes thereof BRACCO INTERNATIONAL B.V. 1997-03-04 US disclosed
EP-0629617-A1 Heteroatom-bearing ligands and metal complexes thereof BRACCO International B.V. (NL) 1994-12-21 EP disclosed