SCHEMBL5314656

SCHEMBL5314656

CC([AsH2])C/C=C/c1cnc2c(ccn2C)c1

nearest known ligand 0.34

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
APP P05067 1/20 0.34
PIK3CB P42338 1/20 0.31
CYP2A6 P11509 1/20 0.31
CHRNA7 P36544 2/20 0.31
CHRNB2 P17787 2/20 0.30
CHRNA4 P43681 2/20 0.30
CACNA1G O43497 1/20 0.30
CACNA1H O95180 1/20 0.30
CACNA1I Q9P0X4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29935942 0.73 CYP2A6 (0.53) APPPIK3CBCYP2A6CHRNA7CACNA1G
SCHEMBL6952609 0.73 CYP2A6 (0.53) APPPIK3CBCYP2A6CHRNA7CACNA1G
SCHEMBL3716346 0.73 APP (0.40) APPPIK3CBCYP2A6CHRNA7CACNA1G
SCHEMBL17173829 0.69 HDAC1 (0.50)
SCHEMBL15218207 0.68 APP (0.41) APPPIK3CBCHRNA7CACNA1GCACNA1H
SCHEMBL12896058 0.68 PIK3CB (0.39) APPPIK3CBCHRNA7CHRNB2CHRNA4
SCHEMBL25150552 0.67 APP (0.38) APPPIK3CBCHRNA7CACNA1GCACNA1H
SCHEMBL17173420 0.67 KDM4E (0.43) APPCHRNA7CACNA1GCACNA1HCACNA1I
Cyanide SCHEMBL22130245 0.67 APP (0.36) APPPIK3CBCYP2A6CHRNA7CACNA1G
SCHEMBL25469510 0.67 GPBAR1 (0.36) APPPIK3CBCHRNA7CACNA1GCACNA1H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1814852-A2 HYDROXYBENZOATE SALTS OF METANICOTINE COMPOUNDS Targacept, Inc. (US) 2007-08-08 EP disclosed
WO-2006053082-A2 HYDROXYBENZOATE SALTS OF METANICOTINE COMPOUNDS TARGACEPT, INC. (US) 2006-05-18 WO disclosed