SCHEMBL5315499

SCHEMBL5315499

O=C(O)C(C(=O)O)C(=O)c1n[nH]c2ncccc12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNA2 P20248 1/20 0.39
CDK2 P24941 1/20 0.39
FLT3 P36888 1/20 0.39
CCNA1 P78396 1/20 0.39
CAMKK2 Q96RR4 1/20 0.37
KDM4E B2RXH2 4/20 0.36
MAPK10 P53779 1/20 0.36
HSD17B10 Q99714 1/20 0.36
MAP2K1 Q02750 1/20 0.36
ALDH1A1 P00352 2/20 0.36
MAPK1 P28482 1/20 0.36
ITGB2 P05107 1/20 0.36
ICAM1 P05362 1/20 0.36
ITGAL P20701 1/20 0.36
GSK3A P49840 1/20 0.35
GSK3B P49841 1/20 0.35
AURKA O14965 1/20 0.35
PARP1 P09874 1/20 0.35
YTHDC1 Q96MU7 1/20 0.35
FEN1 P39748 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5924504 0.86 KDM4E (0.42) FLT3KDM4EMAP2K1ALDH1A1GSK3A
SCHEMBL5924495 0.84 MAP2K1 (0.43) CDK2FLT3KDM4EMAPK10HSD17B10
SCHEMBL17321390 0.83 SMN1; SMN2 (0.41) CCNA2CDK2FLT3CCNA1KDM4E
SCHEMBL29623160 0.82 KDM4E (0.47) CCNA2CDK2FLT3CCNA1CAMKK2
SCHEMBL1048847 0.82 KDM4E (0.47) CCNA2CDK2FLT3CCNA1CAMKK2
SCHEMBL28098788 0.80 MAP2K1 (0.41) CCNA2CDK2FLT3CCNA1CAMKK2
SCHEMBL5924436 0.78 MAP2K1 (0.43) CAMKK2KDM4EMAPK10HSD17B10MAP2K1
SCHEMBL29732854 0.78 CAMKK2 (0.46) CAMKK2KDM4EMAPK10HSD17B10MAP2K1
SCHEMBL5924295 0.78 KDM4E (0.40) CCNA2CDK2FLT3CCNA1CAMKK2
SCHEMBL1384475 0.78 CAMKK2 (0.46) CAMKK2KDM4EMAPK10HSD17B10MAP2K1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1814883-A1 BICYCLIC INHIBITORS OR RHO KINASE Vertex Pharmaceuticals Incorporated (US) 2007-08-08 EP disclosed
WO-2006058120-A1 BICYCLIC INHIBITORS OR RHO KINASE VERTEX PHARMACEUTICALS INCORPORATED (US) 2006-06-01 WO disclosed