SCHEMBL5315533

SCHEMBL5315533

CC(C)(C)Sc1ccccc1C#N

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2C9 P11712 1/20 0.50
CYP2C19 P33261 1/20 0.50
TSHR P16473 1/20 0.46
AR P10275 6/20 0.43
HTT P42858 2/20 0.40
ALDH1A1 P00352 2/20 0.40
XDH P47989 1/20 0.39
LMNA P02545 2/20 0.38
POLB P06746 2/20 0.38
MAPT P10636 2/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
DDB1 Q16531 1/20 0.37
CRBN Q96SW2 1/20 0.37
HSD11B1 P28845 1/20 0.36
GAA P10253 2/20 0.36
PDK1 Q15118 1/20 0.36
PDK2 Q15119 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8715118 0.84 CYP1A2 (0.41) CYP1A2CYP3A4CYP2C9CYP2C19TSHR
SCHEMBL16925204 0.83 CYP1A2 (0.40) CYP1A2CYP3A4CYP2C9CYP2C19TSHR
SCHEMBL16555998 0.78 CYP1A2 (0.50) CYP1A2CYP3A4CYP2C9CYP2C19TSHR
SCHEMBL9018854 0.78 CYP1A2 (0.50) CYP1A2CYP3A4CYP2C9CYP2C19TSHR
SCHEMBL6934720 0.78 AOC3 (0.37) CYP2C19TSHRALDH1A1MAPTMEN1
SCHEMBL514630 0.77 CYP1A2 (0.53) CYP1A2CYP3A4CYP2C9CYP2C19TSHR
SCHEMBL224653 0.77 CYP1A2 (0.57) CYP1A2CYP3A4CYP2C9CYP2C19TSHR
SCHEMBL100732 0.77 CYP1A2 (0.76) CYP1A2CYP3A4CYP2C9CYP2C19TSHR
SCHEMBL30320250 0.77 CYP1A2 (0.57) CYP1A2CYP3A4CYP2C9CYP2C19TSHR
Fluoride SCHEMBL28296217 0.76 CYP1A2 (0.52) CYP1A2CYP3A4CYP2C9CYP2C19TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 38 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112920135-A Dimer impurity in ziprasidone hydrochloride raw material and preparation method thereof 海南鑫开源医药科技有限公司 2021-06-08 CN claimed
CN-108003113-A A kind of synthetic method for treating diabetes medicament 上海工程技术大学 2018-05-08 CN claimed
EP-1081141-B1 Method for producing 1,2-benzisothiazol-3-ones SUMITOMO SEIKA CHEMICALS (JP) 2005-05-04 EP claimed
EP-1081141-A1 Method for producing 1,2-benzisothiazol-3-ones SUMITOMO SEIKA CHEMICALS CO., LTD. (JP) 2001-03-07 EP claimed
EP-0741129-B1 Cyanobenzenesulfenyl halide and process for preparation of 3-substituted benzisothiazole using it SUMITOMO SEIKA CHEMICALS (JP) 1999-06-09 EP claimed
US-5679827-A Cyanobenzenesulfenyl halide and process for preparation of 3-substituted benzisothiazole using the same SUMITOMO SEIKA CHEMICALS CO., LTD. (JP) 1997-10-21 US claimed
EP-0741129-A2 Cyanobenzenesulfenyl halide and process for preparation of 3-substituted benzisothiazole using it SUMITOMO SEIKA CHEMICALS CO., LTD. (JP) 1996-11-06 EP claimed
EP-0702008-A2 Method for producing 1,2-benzisothiazol-3-ones SUMITOMO SEIKA CHEMICALS CO., LTD. (JP) 1996-03-20 EP claimed
CN-108003113-B Synthetic method of medicine for treating diabetes 上海工程技术大学 2021-06-11 CN disclosed
CN-108003113-B Synthetic method of medicine for treating diabetes 上海工程技术大学 2021-06-11 CN disclosed
CN-112920135-A Dimer impurity in ziprasidone hydrochloride raw material and preparation method thereof 海南鑫开源医药科技有限公司 2021-06-08 CN disclosed
CN-108003113-A A kind of synthetic method for treating diabetes medicament 上海工程技术大学 2018-05-08 CN disclosed
CN-108003113-A A kind of synthetic method for treating diabetes medicament 上海工程技术大学 2018-05-08 CN disclosed
US-9346795-B2 Substituted sulfonamides useful as antiapoptotic Bcl inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2016-05-24 US disclosed
US-5773626-A HALOGENATION OF A 2-(ALKYLTHIO)BENZALDEHYDE OXIME SUMITOMO SEIKA CHEMICALS CO., LTD. (JP) 1998-06-30 US disclosed
US-5756806-A Cyanobenzenesulfenyl halide and process for preparation of 3-substituted benzisothiazole using the same SUMITOMO SEIKA CHEMICALS CO., LTD. (JP) 1998-05-26 US disclosed
US-5679827-A Cyanobenzenesulfenyl halide and process for preparation of 3-substituted benzisothiazole using the same SUMITOMO SEIKA CHEMICALS CO., LTD. (JP) 1997-10-21 US disclosed
US-5633384-A FROM O-ALKYLTHIOBENZONITRILES SUMITOMO SEIKA CHEMICALS CO., LTD. (JP) 1997-05-27 US disclosed
EP-0741129-A2 Cyanobenzenesulfenyl halide and process for preparation of 3-substituted benzisothiazole using it SUMITOMO SEIKA CHEMICALS CO., LTD. (JP) 1996-11-06 EP disclosed
EP-0702008-A2 Method for producing 1,2-benzisothiazol-3-ones SUMITOMO SEIKA CHEMICALS CO., LTD. (JP) 1996-03-20 EP disclosed