SCHEMBL5315858

SCHEMBL5315858

NCCCOc1ccc2nccc(NC(=O)O)c2n1.c1cc2c(cc1CNC1CCCCC1)OCCO2

nearest known ligand 0.62

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 12/20 0.62
HSF1 Q00613 1/20 0.40
KDM4E B2RXH2 1/20 0.37
TDP1 Q9NUW8 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5260199 0.89 KCNH2 (0.76) KCNH2
SCHEMBL14498816 0.89 KCNH2 (0.63) KCNH2HSF1
SCHEMBL5260215 0.80 KCNH2 (0.76) KCNH2
SCHEMBL5265007 0.80 KCNH2 (0.63) KCNH2
SCHEMBL5261624 0.78 KCNH2 (0.79) KCNH2
SCHEMBL14498785 0.78 KCNH2 (0.79) KCNH2
SCHEMBL5263867 0.77 KCNH2 (0.56) KCNH2
SCHEMBL5264690 0.76 KCNH2 (0.61) KCNH2
SCHEMBL5262423 0.76 KCNH2 (0.59) KCNH2
SCHEMBL5260170 0.75 KCNH2 (0.55) KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1399443-B1 NITROGEN-CONTAINING BICYCLIC HETEROCYCLES FOR USE AS ANTIBACTERIALS SMITHKLINE BEECHAM PLC (GB) 2007-12-12 EP claimed