SCHEMBL5316565

SCHEMBL5316565

CC(C)(C)OC(=O)N[C@H]1CCC(NC(=O)CNC(=O)c2cccc(C(F)(F)F)c2)C(CN2CCCC2)C1

nearest known ligand 0.56

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 20/20 0.56
CCR3 P51677 1/20 0.52
CYP2D6 P10635 1/20 0.51
KCNH2 Q12809 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5033694 1.00 CCR2 (0.56) CCR2CCR3CYP2D6KCNH2
SCHEMBL5316562 1.00 CCR2 (0.56) CCR2CCR3CYP2D6KCNH2
SCHEMBL5033698 1.00 CCR2 (0.56) CCR2CCR3CYP2D6KCNH2
SCHEMBL5027207 0.86 CCR2 (0.57) CCR2CCR3CYP2D6KCNH2
SCHEMBL5029573 0.85 CCR2 (0.70) CCR2CYP2D6KCNH2
SCHEMBL5029564 0.85 CCR2 (0.70) CCR2CYP2D6KCNH2
SCHEMBL5029659 0.84 CCR2 (0.66) CCR2CYP2D6KCNH2
SCHEMBL5029235 0.83 CCR2 (0.72) CCR2KCNH2
SCHEMBL5029232 0.83 CCR2 (0.72) CCR2KCNH2
SCHEMBL5033978 0.83 CCR2 (0.60) CCR2CCR3CYP2D6KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1656138-A4 SUBSTITUTED CYCLOALKYAMINE DERIVATIVES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY BRISTOL MYERS SQUIBB CO (US) 2007-04-18 EP disclosed
EP-1656138-A2 SUBSTITUTED CYCLOALKYAMINE DERIVATIVES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY Bristol-Myers Squibb Company (US) 2006-05-17 EP disclosed
WO-2005020899-A2 SUBSTITUTED CYCLOALKYAMINE DERIVATIVES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY BRISTOL-MYERS SQUIBB COMPANY (US) 2005-03-10 WO disclosed