SCHEMBL5316745

SCHEMBL5316745

CCOC(=O)c1cc(O)ccc1Br

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 5/20 0.70
CA1 P00915 5/20 0.70
CA2 P00918 5/20 0.70
CA7 P43166 5/20 0.70
CA9 Q16790 5/20 0.70
CA14 Q9ULX7 5/20 0.70
ESR1 P03372 2/20 0.53
ESR2 Q92731 2/20 0.53
TSHR P16473 1/20 0.52
MIF P14174 1/20 0.51
PFKFB3 Q16875 1/20 0.51
MAOA P21397 1/20 0.51
MAOB P27338 1/20 0.51
EGFR P00533 2/20 0.48
NR1H2 P55055 1/20 0.47
NR1H3 Q13133 1/20 0.47
GAA P10253 1/20 0.47
ALOX5 P09917 1/20 0.46
SERPINE1 P05121 1/20 0.46
KDM4E B2RXH2 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22833376 0.86 CA12 (0.70) CA12CA1CA2CA7CA9
SCHEMBL17022287 0.84 ALDH1A1 (0.55) CA12CA1CA2CA7CA9
SCHEMBL30294343 0.84 TSHR (0.53) CA12CA1CA2CA7CA9
SCHEMBL1814266 0.84 TSHR (0.53) CA12CA1CA2CA7CA9
SCHEMBL10449048 0.84 CA12 (0.77) CA12CA1CA2CA7CA9
SCHEMBL4882699 0.83 HPGD (0.56) CA12CA1CA2CA7CA9
SCHEMBL277473 0.83 CA12 (0.57) CA12CA1CA2CA7CA9
SCHEMBL550228 0.82 CA12 (0.74) CA12CA1CA2CA7CA9
SCHEMBL29457603 0.82 CA12 (1.00) CA12CA1CA2CA7CA9
SCHEMBL39259 0.82 CA12 (1.00) CA12CA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9382188-B2 Aromatic ring compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-07-05 US disclosed
EP-2816023-A1 AROMATIC RING COMPOUND Takeda Pharmaceutical Company Limited (JP) 2014-12-24 EP disclosed
WO-2007058504-A1 NOVEL COMPOUNDS AS AGONIST FOR PPAR GAMMA AND PPAR ALPHA, METHOD FOR PREPARATION OF THE SAME, AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME LG LIFE SCIENCES, LTD. (KR) 2007-05-24 WO disclosed