SCHEMBL5318002

SCHEMBL5318002

Cc1nc2sc(C)c(C)c2c(-c2ccccc2)c1CC=O

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.46
RXFP1 Q9HBX9 1/20 0.43
SMN1; SMN2 Q16637 4/20 0.42
KDM4E B2RXH2 2/20 0.42
HPGD P15428 1/20 0.42
ELANE P08246 1/20 0.41
LMNA P02545 1/20 0.39
KMT2A Q03164 2/20 0.39
MEN1 O00255 1/20 0.39
TSHR P16473 1/20 0.39
POLB P06746 1/20 0.38
HTT P42858 1/20 0.37
ATM Q13315 1/20 0.37
ABCB1 P08183 1/20 0.37
MAOB P27338 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4056576 0.85 SMN1; SMN2 (0.40) ALDH1A1RXFP1SMN1; SMN2KDM4EHPGD
SCHEMBL5316508 0.76 ALDH1A1 (0.48) ALDH1A1SMN1; SMN2KDM4EHPGDLMNA
SCHEMBL28661629 0.75 SMN1; SMN2 (0.65) SMN1; SMN2KDM4ELMNAKMT2AMEN1
SCHEMBL4055022 0.74 ALDH1A1 (0.48) ALDH1A1SMN1; SMN2KDM4EHPGDLMNA
SCHEMBL99422 0.73 KMT2A (0.65) SMN1; SMN2KDM4ELMNAKMT2APOLB
SCHEMBL4057323 0.72 MAPT (0.44) ALDH1A1RXFP1SMN1; SMN2KDM4EHPGD
SCHEMBL5343442 0.70 ALDH1A1 (0.44) ALDH1A1RXFP1SMN1; SMN2KDM4EHPGD
SCHEMBL5177389 0.68 KDM4E (0.52) ALDH1A1RXFP1SMN1; SMN2KDM4ELMNA
SCHEMBL99707 0.68 KMT2A (0.51) ALDH1A1KDM4EELANEKMT2A
SCHEMBL5177676 0.68 SMN1; SMN2 (0.54) ALDH1A1SMN1; SMN2KDM4ELMNAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1828199-A1 THIENO-PYRIDINE DERIVATIVES AS GABA-B ALLOSTERIC ENHANCERS F. Hoffmann-Roche AG (CH) 2007-09-05 EP claimed
WO-2006063732-A1 THIENO-PYRIDINE DERIVATIVES AS GABA-B ALLOSTERIC ENHANCERS F.HOFFMANN-LA ROCHE AG (CH) 2006-06-22 WO claimed
EP-1828199-A1 THIENO-PYRIDINE DERIVATIVES AS GABA-B ALLOSTERIC ENHANCERS F. Hoffmann-Roche AG (CH) 2007-09-05 EP disclosed
WO-2006063732-A1 THIENO-PYRIDINE DERIVATIVES AS GABA-B ALLOSTERIC ENHANCERS F.HOFFMANN-LA ROCHE AG (CH) 2006-06-22 WO disclosed