SCHEMBL5318403

SCHEMBL5318403

Cc1c[nH]c2nccc(Nc3ccc(Nc4nc(N)cc(C(F)(F)F)n4)cc3F)c12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 10/20 0.47
CYP3A4 P08684 4/20 0.47
AURKA O14965 3/20 0.41
CDC7 O00311 1/20 0.41
CHEK1 O14757 1/20 0.41
PDPK1 O15530 1/20 0.41
DAPK3 O43293 1/20 0.41
DYRK3 O43781 1/20 0.41
CACNA1F O60840 1/20 0.41
RAF1 P04049 1/20 0.41
ERBB2 P04626 1/20 0.41
NTRK1 P04629 1/20 0.41
INSR P06213 1/20 0.41
CDK1 P06493 1/20 0.41
FES P07332 1/20 0.41
CSF1R P07333 1/20 0.41
LYN P07948 1/20 0.41
MET P08581 1/20 0.41
ROS1 P08922 1/20 0.41
KIT P10721 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8272279 0.86 ROCK2 (0.56) ROCK2CYP3A4AURKACDC7CHEK1
SCHEMBL2887314 0.79 ROCK2 (0.54) ROCK2CYP3A4AURKACDC7CHEK1
SCHEMBL2886218 0.77 ROCK2 (0.44) ROCK2CYP3A4AURKACDC7CHEK1
SCHEMBL2881276 0.76 ROCK2 (0.71) ROCK2CYP3A4AURKACDC7CHEK1
SCHEMBL8270531 0.73 ROCK2 (0.73) ROCK2CYP3A4AURKACDC7CHEK1
SCHEMBL2884975 0.73 ROCK2 (0.39) ROCK2CYP3A4AURKACDC7CHEK1
SCHEMBL5097939 0.72 ROCK2 (0.61) ROCK2CYP3A4AURKACDC7CHEK1
SCHEMBL8283424 0.72 ROCK2 (0.77) ROCK2CYP3A4AURKACDC7CHEK1
SCHEMBL2887689 0.69 ROCK2 (0.56) ROCK2CYP3A4AURKACDC7CHEK1
SCHEMBL2881782 0.69 ROCK2 (0.45) ROCK2CYP3A4AURKACDC7CHEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1742945-A1 SUBSTITUTED PHENYLAMINO-PYRIMIDINES Bayer HealthCare AG (DE) 2007-01-17 EP disclosed
WO-2005108397-A1 SUBSTITUTED PHENYLAMINO-PYRIMIDINES BAYER HEALTHCARE AG (DE) 2005-11-17 WO disclosed