SCHEMBL5318644

SCHEMBL5318644

Nc1ncc(-c2cccc(C(F)(F)F)c2)cn1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 2/20 0.60
ADORA1 P30542 2/20 0.60
MAP4K4 O95819 1/20 0.59
ALDH1A1 P00352 3/20 0.55
GAA P10253 1/20 0.55
ATM Q13315 1/20 0.55
L3MBTL1 Q9Y468 1/20 0.52
PIK3CB P42338 1/20 0.52
SCN2A Q99250 2/20 0.51
PARP1 P09874 1/20 0.51
TSHR P16473 1/20 0.50
MAPK1 P28482 1/20 0.50
HRH1 P35367 1/20 0.50
HRH4 Q9H3N8 1/20 0.50
CCNT1 O60563 1/20 0.49
CCNA2 P20248 1/20 0.49
CDK2 P24941 1/20 0.49
CDK9 P50750 1/20 0.49
IDO1 P14902 1/20 0.49
KDM4E B2RXH2 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17362398 0.84 ADORA2A (0.59) ADORA2AADORA1PIK3CBSCN2AHRH1
SCHEMBL30704262 0.83 MAP4K4 (0.62) ADORA2AADORA1MAP4K4ALDH1A1GAA
SCHEMBL28051302 0.83 MAP4K4 (0.62) ADORA2AADORA1MAP4K4ALDH1A1GAA
SCHEMBL12449552 0.82 MAP4K4 (0.59) ADORA2AADORA1MAP4K4ALDH1A1GAA
SCHEMBL11483670 0.82 ALDH1A1 (0.56) ADORA2AADORA1ALDH1A1GAAATM
SCHEMBL28307660 0.81 PARP1 (0.51) ADORA2AADORA1ALDH1A1GAAATM
SCHEMBL29636028 0.81 PARP1 (0.51) ADORA2AADORA1ALDH1A1GAAATM
SCHEMBL29678302 0.80 TSHR (0.58) ALDH1A1SCN2ATSHRMAPK1IDO1
SCHEMBL1263144 0.80 TSHR (0.58) ALDH1A1SCN2ATSHRMAPK1IDO1
SCHEMBL29655536 0.79 ADORA2A (0.72) ADORA2AADORA1SCN2ACCNT1CCNA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007096764-A2 BICYCLIC HETEROARYL DERIVATIVES AS CANNABINOID RECEPTOR MODULATORS GLENMARK PHARMACEUTICALS S.A. (US) 2007-08-30 WO claimed
WO-2022195522-A1 INHIBITORS OF ANO6 AND THEIR USES THEREOF ILDONG PHARMACEUTICAL CO., LTD. (KR) 2022-09-22 WO disclosed
WO-2022157686-A1 INHIBITORS OF ANOCTAMIN 6 PROTEIN AND USES THEREOF ILDONG PHARMACEUTICAL CO., LTD. (KR) 2022-07-28 WO disclosed
WO-2007096764-A2 BICYCLIC HETEROARYL DERIVATIVES AS CANNABINOID RECEPTOR MODULATORS GLENMARK PHARMACEUTICALS S.A. (US) 2007-08-30 WO disclosed