SCHEMBL531912

SCHEMBL531912

C[C@@H]1[C@@H](c2cc(C(F)(F)F)cc(C(F)(F)F)c2)OC(=O)N1Cc1cc(C(F)(F)F)ccc1I

nearest known ligand 0.61

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CETP P11597 16/20 0.61
NR1I2 O75469 3/20 0.61
PTGDR2 Q9Y5Y4 4/20 0.56
KCNH2 Q12809 2/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL532579 1.00 CETP (0.61) CETPNR1I2PTGDR2KCNH2
SCHEMBL531911 1.00 CETP (0.61) CETPNR1I2PTGDR2KCNH2
SCHEMBL14874761 1.00 CETP (0.61) CETPNR1I2PTGDR2KCNH2
SCHEMBL3577311 1.00 CETP (0.61) CETPNR1I2PTGDR2KCNH2
SCHEMBL12696971 0.94 CETP (0.55) CETPNR1I2PTGDR2KCNH2
SCHEMBL1529173 0.93 CETP (0.54) CETPNR1I2PTGDR2KCNH2
SCHEMBL4307662 0.90 CETP (0.55) CETPNR1I2PTGDR2KCNH2
SCHEMBL1529174 0.89 CETP (0.50) CETPNR1I2PTGDR2
SCHEMBL531641 0.88 CETP (0.51) CETPNR1I2
SCHEMBL531640 0.88 CETP (0.51) CETPNR1I2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2029560-B1 1,3-OXAZOLIDIN-2-ONE DERIVATIVES USEEFUL AS CETP INHIBITORS MERCK SHARP & DOHME (US) 2013-04-24 EP disclosed
EP-2415759-A1 CETP inhibitors Merck Sharp & Dohme Corporation (US) 2012-02-08 EP disclosed