SCHEMBL5320022

SCHEMBL5320022

CN1CCC(N(C)C(=O)c2ccc3c(c2)nc(N2CCCC2)n3C)CC1

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 1/20 0.49
ADORA1 P30542 1/20 0.49
POLB P06746 1/20 0.47
TLR9 Q9NR96 1/20 0.45
TLR8 Q9NR97 1/20 0.45
TLR7 Q9NYK1 1/20 0.45
HDAC6 Q9UBN7 2/20 0.45
HRH3 Q9Y5N1 1/20 0.45
ITK Q08881 7/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
MRGPRX2 Q96LB1 3/20 0.43
CNR2 P34972 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5316323 0.86 ITK (0.48) POLBHDAC6HRH3ITKCNR2
SCHEMBL5317398 0.80 ITK (0.49) ITKMRGPRX2CNR2
SCHEMBL5318430 0.80 ITK (0.49) HRH3ITKCNR2
SCHEMBL5315622 0.80 TLR9 (0.46) ADORA2AADORA1TLR9TLR8TLR7
SCHEMBL5315400 0.79 FLT3 (0.48) TLR9TLR8TLR7ITK
SCHEMBL5320783 0.79 ITK (0.47) ITKMRGPRX2
SCHEMBL5316334 0.78 CNR2 (0.52) ITKCNR2
SCHEMBL4258690 0.78 HDAC6 (0.53) POLBHDAC6MEN1KMT2A
SCHEMBL5317039 0.78 ITK (0.46) HDAC6HRH3ITKCNR2
SCHEMBL5316556 0.78 HDAC6 (0.63) ADORA2AADORA1HDAC6HRH3ITK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007069053-A1 BENZIMIDAZOLE ANTAGONISTS OF THE H-3 RECEPTOR PFIZER PRODUCTS INC. (US) 2007-06-21 WO claimed
WO-2007069053-A1 BENZIMIDAZOLE ANTAGONISTS OF THE H-3 RECEPTOR PFIZER PRODUCTS INC. (US) 2007-06-21 WO disclosed