SCHEMBL532004

SCHEMBL532004

CC1Oc2ccc(OC3CCN(C(=O)O)CC3)cc2NC1=O

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SMYD3 Q9H7B4 3/20 0.46
PARP1 P09874 8/20 0.45
HTR1A P08908 2/20 0.41
HTR7 P34969 2/20 0.41
KCNH2 Q12809 1/20 0.41
HRH3 Q9Y5N1 5/20 0.41
PDE3B Q13370 2/20 0.40
PDE3A Q14432 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10222934 0.87 HRH3 (0.53) SMYD3PARP1HRH3
SCHEMBL532300 0.82 PARP1 (0.47) SMYD3PARP1HTR1AHTR7KCNH2
SCHEMBL4185512 0.80 HTR1A (0.55) PARP1HTR1A
SCHEMBL23842802 0.80 PARP1 (0.50) SMYD3PARP1HTR1AHTR7KCNH2
SCHEMBL532182 0.80 PARP1 (0.65) SMYD3PARP1
SCHEMBL533459 0.78 PARP1 (0.51) SMYD3PARP1HTR1AHTR7KCNH2
SCHEMBL531980 0.78 SMYD3 (0.59) SMYD3PARP1HRH3
SCHEMBL23830906 0.78 HRH3 (0.42) SMYD3PARP1HTR1AHTR7KCNH2
SCHEMBL532159 0.77 PARP1 (0.68) SMYD3PARP1
SCHEMBL4196161 0.74 HTR1A (0.51) PARP1HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8669249-B2 Poly (ADP-ribose) polymerase (PARP) inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2014-03-11 US disclosed
US-20120094992-A1 POLY (ADP-RIBOSE) POLYMERASE (PARP) INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-04-19 US disclosed
EP-2415767-A1 Poly (ADP-ribose) Polymerase (PARP) Inhibitors Takeda Pharmaceutical Company Limited (JP) 2012-02-08 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120094992-A1 POLY (ADP-RIBOSE) POLYMERASE (PARP) INHIBITORS PARP1, PARP2, PARP3 SMYD3 3712/4885PARP1 1/4885HTR1A 2476/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.