SCHEMBL5320569

SCHEMBL5320569

COc1ccc(N2CCN(C)CC2)c2[nH]c(C(=O)O)cc(=O)c12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.46
HPGD P15428 3/20 0.46
HRH4 Q9H3N8 2/20 0.42
HTR1B P28222 7/20 0.42
HTR1A P08908 5/20 0.41
HTR1D P28221 5/20 0.41
ALDH1A1 P00352 2/20 0.40
DRD2 P14416 2/20 0.40
DRD3 P35462 2/20 0.40
TSHR P16473 1/20 0.40
CASP1 P29466 1/20 0.40
CASP7 P55210 1/20 0.40
HTR6 P50406 3/20 0.40
HTR2A P28223 2/20 0.40
HTR2C P28335 2/20 0.40
HTR7 P34969 1/20 0.40
ERAP1 Q9NZ08 2/20 0.39
GPR35 Q9HC97 1/20 0.39
LMNA P02545 1/20 0.39
DRD4 P21917 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5340176 0.86 KDM4E (0.39) KDM4EHPGDHRH4HTR1BHTR1A
SCHEMBL5322764 0.84 HRH4 (0.45) KDM4EHRH4HTR1BALDH1A1DRD2
SCHEMBL14437521 0.79 HTR1B (0.49) KDM4EHTR1BHTR1AHTR1DALDH1A1
SCHEMBL5322699 0.79 HTR1B (0.58) HTR1BHTR1AHTR1DALDH1A1TSHR
SCHEMBL14437529 0.79 HTR1B (0.58) HPGDHTR1BHTR1AHTR1DALDH1A1
SCHEMBL14437397 0.77 HTR1B (0.57) KDM4EHPGDHTR1BHTR1AHTR1D
SCHEMBL14437524 0.77 HTR1B (0.56) HPGDHTR1BHTR1AHTR1DALDH1A1
SCHEMBL14437849 0.77 HTR1B (0.56) HTR1BHTR1AHTR1DALDH1A1TSHR
SCHEMBL14437526 0.76 HTR1B (0.46) KDM4EHTR1BHTR1AHTR1DALDH1A1
SCHEMBL4988681 0.76 HTR1B (0.63) KDM4EHPGDHRH4HTR1BALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007097697-A1 THERAPEUTIC QUINOLINE COMPOUNDS THAT ARE 5HT1B MODULATORS ASTRAZENECA AB (SE) 2007-08-30 WO claimed
WO-2007097697-A1 THERAPEUTIC QUINOLINE COMPOUNDS THAT ARE 5HT1B MODULATORS ASTRAZENECA AB (SE) 2007-08-30 WO disclosed