SCHEMBL5320870

SCHEMBL5320870

COc1cc2c(cc1C)NC(=O)N(C(C)C)N=C2C1CCCCC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 8/20 0.42
PDE4A P27815 7/20 0.42
PDE4C Q08493 7/20 0.42
PDE4D Q08499 7/20 0.42
PTH1R Q03431 2/20 0.35
HTR2A P28223 1/20 0.34
HTT P42858 2/20 0.33
CHRM1 P11229 1/20 0.33
PDE3B Q13370 1/20 0.32
PDE3A Q14432 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
MCOLN3 Q8TDD5 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
PDE10A Q9Y233 1/20 0.32
PDE7A Q13946 1/20 0.32
TNKS O95271 1/20 0.31
TNKS2 Q9H2K2 1/20 0.31
KDM4E B2RXH2 1/20 0.31
USP2 O75604 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5352183 0.84 PTH1R (0.36) PDE4BPDE4APDE4CPDE4DPTH1R
SCHEMBL5351487 0.83 PTH1R (0.36) PDE4BPDE4APDE4CPDE4DPTH1R
SCHEMBL5354276 0.82 PTH1R (0.34) PDE4BPDE4APDE4CPDE4DPTH1R
SCHEMBL5361939 0.81 PDE4A (0.40) PDE4BPDE4APDE4CPDE4DPTH1R
SCHEMBL5325236 0.80 PTH1R (0.46) PDE4BPDE4APDE4CPDE4DPTH1R
SCHEMBL5349032 0.76 PTH1R (0.49) PDE4BPDE4APDE4CPDE4DPTH1R
SCHEMBL5326236 0.76 PTH1R (0.41) PTH1R
SCHEMBL5326300 0.72 PTH1R (0.48) PDE4BPDE4APDE4CPDE4DPTH1R
SCHEMBL5345828 0.71 PTH1R (0.47) PDE4BPDE4APDE4CPDE4DPTH1R
SCHEMBL5323094 0.70 PDE4B (0.39) PDE4BPDE4APDE4CPDE4DHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006129120-A9 BENZOTRIAZEPINONE DERIVATIVES JAMES BLACK FOUNDATION (GB) 2007-03-22 WO disclosed
WO-2006129120-A2 BENZOTRIAZEPINONE DERIVATIVES JAMES BLACK FOUNDATION (GB) 2006-12-07 WO disclosed