SCHEMBL5320900

SCHEMBL5320900

COc1cccc(-c2cnc3nc(-c4ccccc4)c(-c4ccc(Cl)cc4Cl)n3c2)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 6/20 0.52
DPP8 Q6V1X1 4/20 0.52
DPP9 Q86TI2 3/20 0.52
AKT1 P31749 2/20 0.43
AKT2 P31751 2/20 0.43
GRM5 P41594 1/20 0.43
ADORA2A P29274 1/20 0.43
ADORA1 P30542 1/20 0.43
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2C19 P33261 1/20 0.42
KMT2A Q03164 1/20 0.40
SLC2A1 P11166 1/20 0.40
PIK3CA P42336 1/20 0.40
PIK3CB P42338 1/20 0.40
PIK3CG P48736 1/20 0.40
MAPT P10636 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
BACE1 P56817 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5320273 0.96 DPP4 (0.52) DPP4DPP8DPP9AKT1AKT2
SCHEMBL5337653 0.93 DPP4 (0.49) DPP4DPP8DPP9AKT1AKT2
SCHEMBL5321406 0.86 AKT1 (0.49) DPP4DPP8DPP9AKT1AKT2
SCHEMBL5318881 0.82 DPP4 (0.48) DPP4DPP8DPP9AKT1AKT2
Hydrochloric Acid SCHEMBL5344135 0.82 DPP4 (0.47) DPP4DPP8DPP9AKT1AKT2
SCHEMBL5336486 0.81 AKT1 (0.39) DPP4DPP8DPP9AKT1AKT2
SCHEMBL5344598 0.80 KMT2A (0.53) DPP4DPP8DPP9AKT1AKT2
SCHEMBL5352678 0.79 AKT1 (0.43) DPP4DPP8DPP9AKT1AKT2
SCHEMBL5341559 0.79 DPP4 (0.45) DPP4DPP8DPP9AKT1AKT2
SCHEMBL5321252 0.78 DPP4 (0.54) DPP4DPP8DPP9ADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007096764-A2 BICYCLIC HETEROARYL DERIVATIVES AS CANNABINOID RECEPTOR MODULATORS GLENMARK PHARMACEUTICALS S.A. (US) 2007-08-30 WO claimed
WO-2007096764-A2 BICYCLIC HETEROARYL DERIVATIVES AS CANNABINOID RECEPTOR MODULATORS GLENMARK PHARMACEUTICALS S.A. (US) 2007-08-30 WO disclosed