SCHEMBL5344598

SCHEMBL5344598

COc1ccc(-c2c(-c3ccc(Cl)cc3)nc3ncc(-c4cccc(Cl)c4)cn23)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.53
AKT1 P31749 4/20 0.48
AKT2 P31751 4/20 0.48
MGAM O43451 2/20 0.42
GAA P10253 2/20 0.42
SI P14410 2/20 0.42
MGAM2 Q2M2H8 2/20 0.42
ALDH1A1 P00352 3/20 0.41
MEN1 O00255 1/20 0.41
USP2 O75604 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C19 P33261 1/20 0.41
RECQL P46063 1/20 0.41
RAB9A P51151 3/20 0.41
NPC1 O15118 2/20 0.41
KDM4E B2RXH2 2/20 0.41
SLC2A1 P11166 1/20 0.40
NR1I3 Q14994 1/20 0.40
MAOB P27338 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5321406 0.91 AKT1 (0.49) KMT2AAKT1AKT2ALDH1A1USP2
SCHEMBL5325683 0.91 AKT1 (0.51) KMT2AAKT1AKT2GAAALDH1A1
SCHEMBL5343644 0.88 GRIN1 (0.46) KMT2AAKT1AKT2MGAMGAA
SCHEMBL5342012 0.85 AKT1 (0.44) KMT2AAKT1AKT2GAAALDH1A1
SCHEMBL5320273 0.84 DPP4 (0.52) KMT2AAKT1AKT2MEN1CYP1A2
SCHEMBL5345880 0.83 PTGS2 (0.55) AKT1AKT2NR1I3
SCHEMBL5349048 0.83 AKT1 (0.48) KMT2AAKT1AKT2GAAALDH1A1
SCHEMBL5341386 0.82 AKT1 (0.49) AKT1AKT2GAAALDH1A1RAB9A
SCHEMBL5322231 0.81 AKT1 (0.48) AKT1AKT2GAAALDH1A1CYP1A2
SCHEMBL5352678 0.81 AKT1 (0.43) KMT2AAKT1AKT2GAAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007096764-A2 BICYCLIC HETEROARYL DERIVATIVES AS CANNABINOID RECEPTOR MODULATORS GLENMARK PHARMACEUTICALS S.A. (US) 2007-08-30 WO claimed
WO-2007096764-A2 BICYCLIC HETEROARYL DERIVATIVES AS CANNABINOID RECEPTOR MODULATORS GLENMARK PHARMACEUTICALS S.A. (US) 2007-08-30 WO disclosed