SCHEMBL532302

SCHEMBL532302

C[C@@H]([C@H](O)c1cc(F)cc(F)c1)N(Cc1ccccc1)C(=O)O

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.47
KMT2A Q03164 4/20 0.47
TRPM8 Q7Z2W7 3/20 0.41
NR1I2 O75469 2/20 0.41
HPGD P15428 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
SCN5A Q14524 1/20 0.40
SCN9A Q15858 1/20 0.40
GAA P10253 1/20 0.40
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
POLB P06746 1/20 0.39
HSD17B10 Q99714 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL532301 1.00 MEN1 (0.47) MEN1KMT2ATRPM8NR1I2HPGD
SCHEMBL1529186 0.81 CYP3A4 (0.47) MEN1KMT2ATRPM8HPGDGAA
SCHEMBL1529187 0.81 CYP3A4 (0.47) MEN1KMT2ATRPM8HPGDGAA
SCHEMBL531673 0.79 MEN1 (0.48) MEN1KMT2AHPGDGAAALDH1A1
SCHEMBL531674 0.79 MEN1 (0.48) MEN1KMT2AHPGDGAAALDH1A1
SCHEMBL15670729 0.77 KMT2A (0.59) MEN1KMT2AHPGDALDH1A1LMNA
SCHEMBL15670960 0.77 KMT2A (0.59) MEN1KMT2AHPGDALDH1A1LMNA
SCHEMBL1529072 0.76 CASR (0.49) TRPM8ALDH1A1L3MBTL1
SCHEMBL1529070 0.76 CASR (0.49) TRPM8ALDH1A1L3MBTL1
SCHEMBL531228 0.76 MEN1 (0.48) MEN1KMT2ATRPM8NR1I2TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2415759-A1 CETP inhibitors Merck Sharp & Dohme Corporation (US) 2012-02-08 EP disclosed