SCHEMBL532458

SCHEMBL532458

COc1cc(-c2nn3c(-c4cnc([AsH2])c(C(F)(F)F)c4)cnc3s2)ccc1OC1CCNCC1

nearest known ligand 0.71

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 12/20 0.71
FYN P06241 5/20 0.43
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
HPGD P15428 1/20 0.43
HIF1A Q16665 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2122734 0.91 PIK3CA (0.76) PIK3CAFYNKDM4EALDH1A1HPGD
SCHEMBL532459 0.85 PIK3CA (0.53) PIK3CAKDM4EALDH1A1HPGDHIF1A
SCHEMBL2121448 0.83 PIK3CA (1.00) PIK3CAFYNKDM4EALDH1A1HPGD
SCHEMBL2122629 0.83 PIK3CA (0.80) PIK3CAFYNKDM4EALDH1A1HPGD
SCHEMBL532219 0.79 PIK3CA (0.82) PIK3CAFYNKDM4E
SCHEMBL2122737 0.77 PIK3CA (0.58) PIK3CA
SCHEMBL3714191 0.77 PIK3CA (0.85) PIK3CAFYNKDM4EALDH1A1HPGD
SCHEMBL532710 0.76 PIK3CA (0.58) PIK3CA
SCHEMBL15975810 0.76 PIK3CA (0.73) PIK3CAFYNKDM4EALDH1A1HPGD
SCHEMBL2616030 0.75 PIK3CA (0.49) PIK3CAFYN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2414369-A1 IMIDAZO [2, 1-B][ 1, 3, 4]THIADIAZOLE DERIVATIVES Centro Nacional de Investigaciones Oncológicas (CNIO) (ES) 2012-02-08 EP disclosed
WO-2010112874-A1 IMIDAZO [2, 1-B] [ 1, 3, 4 ] THIADIAZOLE DERIVATIVES CENTRO NACIONAL DE INVESTIGACIONES ONCOLOGICAS (CNIO) (ES) 2010-10-07 WO disclosed