SCHEMBL532459

SCHEMBL532459

COc1cc(-c2nn3cc(-c4cnc([AsH2])c(C(F)(F)F)c4)nc3s2)ccc1OC1CCNCC1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 7/20 0.53
F2RL3 Q96RI0 6/20 0.42
CTSS P25774 1/20 0.40
CTSK P43235 1/20 0.40
KDM4E B2RXH2 2/20 0.38
ALDH1A1 P00352 2/20 0.38
HPGD P15428 2/20 0.38
HIF1A Q16665 1/20 0.38
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
MAPK1 P28482 1/20 0.36
CYP2C19 P33261 1/20 0.36
HSD17B10 Q99714 1/20 0.36
PIK3CD O00329 1/20 0.35
PIK3CB P42338 1/20 0.35
PIK3CG P48736 1/20 0.35
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2122737 0.92 PIK3CA (0.58) PIK3CAF2RL3CTSSCTSKPIK3CD
SCHEMBL532458 0.85 PIK3CA (0.71) PIK3CAKDM4EALDH1A1HPGDHIF1A
SCHEMBL2122634 0.84 PIK3CA (0.59) PIK3CAF2RL3KDM4EALDH1A1HPGD
SCHEMBL2121456 0.84 PIK3CA (0.71) PIK3CAKDM4EALDH1A1HPGDHIF1A
SCHEMBL532220 0.80 PIK3CA (0.59) PIK3CAF2RL3KDM4EALDH1A1HPGD
SCHEMBL532711 0.78 PIK3CA (0.44) PIK3CAF2RL3PIK3CDPIK3CBPIK3CG
SCHEMBL2122734 0.78 PIK3CA (0.76) PIK3CAKDM4EALDH1A1HPGDHIF1A
SCHEMBL532281 0.75 PIK3CA (0.72) PIK3CAF2RL3KDM4EALDH1A1HPGD
SCHEMBL532218 0.73 TGFBR1 (0.46) PIK3CAKDM4EALDH1A1HPGDCYP1A2
SCHEMBL532581 0.72 PIK3CA (0.59) PIK3CAF2RL3KDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2414369-A1 IMIDAZO [2, 1-B][ 1, 3, 4]THIADIAZOLE DERIVATIVES Centro Nacional de Investigaciones Oncológicas (CNIO) (ES) 2012-02-08 EP disclosed
WO-2010112874-A1 IMIDAZO [2, 1-B] [ 1, 3, 4 ] THIADIAZOLE DERIVATIVES CENTRO NACIONAL DE INVESTIGACIONES ONCOLOGICAS (CNIO) (ES) 2010-10-07 WO disclosed