SCHEMBL532765

SCHEMBL532765

COc1ccc(OC(=O)c2ccc(Cl)cc2)cc1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.70
KMT2A Q03164 6/20 0.64
SMN1; SMN2 Q16637 2/20 0.64
MEN1 O00255 2/20 0.64
CYP1A2 P05177 2/20 0.64
CYP2C9 P11712 2/20 0.64
CYP2C19 P33261 2/20 0.64
LMNA P02545 1/20 0.64
NPC1 O15118 2/20 0.62
RAB9A P51151 2/20 0.62
MAPT P10636 2/20 0.61
CA1 P00915 1/20 0.60
CA2 P00918 1/20 0.60
GFER P55789 1/20 0.59
PRSS1 P07477 1/20 0.59
ACR P10323 1/20 0.59
CYP11B1 P15538 1/20 0.59
CYP11B2 P19099 1/20 0.59
ALDH1A1 P00352 1/20 0.57
CYP3A4 P08684 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL349467 1.00 HPGD (0.70) HPGDKMT2ASMN1; SMN2MEN1CYP1A2
SCHEMBL7591660 0.90 LMNA (0.75) KMT2ASMN1; SMN2MEN1CYP1A2CYP2C9
SCHEMBL12608584 0.90 LMNA (0.75) KMT2ASMN1; SMN2MEN1CYP1A2CYP2C9
SCHEMBL28003430 0.90 KMT2A (0.69) HPGDKMT2ASMN1; SMN2MEN1CYP1A2
SCHEMBL610755 0.90 KMT2A (0.69) HPGDKMT2ASMN1; SMN2MEN1CYP1A2
SCHEMBL12633724 0.90 LMNA (0.75) KMT2ASMN1; SMN2MEN1CYP1A2CYP2C9
SCHEMBL9683516 0.90 KMT2A (0.69) HPGDKMT2ASMN1; SMN2MEN1CYP1A2
SCHEMBL9666088 0.90 LMNA (0.75) KMT2ASMN1; SMN2MEN1CYP1A2CYP2C9
SCHEMBL10599787 0.90 KMT2A (0.69) HPGDKMT2ASMN1; SMN2MEN1CYP1A2
SCHEMBL14393071 0.89 KMT2A (0.69) HPGDKMT2ASMN1; SMN2MEN1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 45 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1511713-B8 COMPOUNDS THAT ABROGATE DNA-DAMAGE-INDUCED CELL CYCLE G2 CHECKPOINT AND/OR AUGMENT THE ANTI-CANCER ACTIVITY OF DNA-DAMAGING TREATMENTS CANBAS CO LTD (JP) 2012-02-08 EP claimed
EP-1511713-B1 COMPOUNDS THAT ABROGATE DNA-DAMAGE-INDUCED CELL CYCLE G2 CHECKPOINT AND/OR AUGMENT THE ANTI-CANCER ACTIVITY OF DNA-DAMAGING TREATMENTS CANBAS CO LTD (JP) 2011-08-17 EP claimed
US-7652042-B2 Compounds that abrogate DNA damage induced cell cycle G2 checkpoint and/or augment anti-cancer activity of DNA-damaging treatments CANBAS CO., LTD. (JP) 2010-01-26 US claimed
US-7629364-B2 Compounds that abrogate DNA-damage-induced cell cycle G2 checkpoint and/or augment anti-cancer activity of DNA-damaging treatments CANBAS CO., LTD. (JP) 2009-12-08 US claimed
US-20080293137-A1 COMPOUNDS THAT ABROGATE DNA DAMAGE INDUCED CELL CYCLE G2 CHECKPOINT AND/OR AUGMENT ANTI-CANCER ACTIVITY OF DNA-DAMAGING TREATMENTS CANBAS CO., LTD. (JP) 2008-11-27 US claimed
US-20080227827-A1 COMPOUNDS THAT ABROGATE DNA DAMAGE INDUCED CELL CYCLE G2 CHECKPOINT AND/OR AUGMENT ANTI-CANCER ACTIVITY OF DNA-DAMAGING TREATMENTS CANBAS CO., LTD. (JP) 2008-09-18 US claimed
US-7407985-B2 Compounds that abrogate DNA damage induced cell cycle G2 checkpoint and/or augment anti-cancer activity of DNA-damaging treatments CANBAS CO., LTD. (JP) 2008-08-05 US claimed
JP-2007501608-A 2007-02-01 JP claimed
US-20060122269-A1 Compounds that abrogate DNA damage induced cell cycle G2 checkpoint and/or augment anti-cancer activity of DNA-damaging treatments CANBAS CO., LTD. (JP) 2006-06-08 US claimed
EP-1664340-A1 SENSITIVITY TEST TO PREDICT EFFICACY OF ANTI-CANCER THERAPIES Canbas Co., Ltd. (JP) 2006-06-07 EP claimed
US-7030111-B2 Compounds that abrogate DNA-damage-induced cell cycle G2 checkpoint and/or augment the anti-cancer activity of DNA damaging treatments CANBAS CO., LTD. (JP) 2006-04-18 US claimed
US-20060014157-A1 Sensitivity test to predict efficacy of anti-cancer therapies CANBAS CO., LTD. (JP) 2006-01-19 US claimed
EP-1511713-A2 COMPOUNDS THAT ABROGATE DNA-DAMAGE-INDUCED CELL CYCLE G2 CHECKPOINT AND/OR AUGMENT THE ANTI-CANCER ACTIVITY OF DNA-DAMAGING TREATMENTS Canbas Co. Ltd. (JP) 2005-03-09 EP claimed
WO-2005014856-A1 SENSITIVITY TEST TO PREDICT EFFICACY OF ANTI-CANCER THERAPIES CANBAS CO., LTD. (JP) 2005-02-17 WO claimed
US-20040198727-A1 Compounds that abrogate DNA-damage-induced cell cycle G2 checkpoint and/or augment the anti-cancer activity of DNA damaging treatments CANBAS CO., LTD. (JP) 2004-10-07 US claimed
WO-2003104181-A2 COMPOUNDS THAT ABROGATE DNA-DAMAGE-INDUCED CELL CYCLE G2 CHECKPOINT AND/OR AUGMENT THE ANTI-CANCER ACTIVITY OF DNA-DAMAGING TREATMENTS CANBAS CO. LTD. (JP) 2003-12-18 WO claimed
EP-1511713-B8 COMPOUNDS THAT ABROGATE DNA-DAMAGE-INDUCED CELL CYCLE G2 CHECKPOINT AND/OR AUGMENT THE ANTI-CANCER ACTIVITY OF DNA-DAMAGING TREATMENTS CANBAS CO LTD (JP) 2012-02-08 EP disclosed
EP-1511713-B1 COMPOUNDS THAT ABROGATE DNA-DAMAGE-INDUCED CELL CYCLE G2 CHECKPOINT AND/OR AUGMENT THE ANTI-CANCER ACTIVITY OF DNA-DAMAGING TREATMENTS CANBAS CO LTD (JP) 2011-08-17 EP disclosed
WO-2003104181-A2 COMPOUNDS THAT ABROGATE DNA-DAMAGE-INDUCED CELL CYCLE G2 CHECKPOINT AND/OR AUGMENT THE ANTI-CANCER ACTIVITY OF DNA-DAMAGING TREATMENTS CANBAS CO. LTD. (JP) 2003-12-18 WO disclosed
US-4612386-A Process for making esters THE DOW CHEMICAL COMPANY (US) 1986-09-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080293137-A1 COMPOUNDS THAT ABROGATE DNA DAMAGE INDUCED CELL CYCLE G2 CHECKPOINT AND/OR AUGMENT ANTI-CANCER ACTIVITY OF DNA-DAMAGING TREATMENTS CDC25C, CHEK1, CDC25A HPGD 1650/4885KMT2A 883/4885SMN1; SMN2 4247/4885
US-20040198727-A1 Compounds that abrogate DNA-damage-induced cell cycle G2 checkpoint and/or augment the anti-cancer activity of DNA damaging treatments CDC25C, CHEK1, DDB1 HPGD 1649/4885KMT2A 766/4885SMN1; SMN2 4352/4885
US-20080227827-A1 COMPOUNDS THAT ABROGATE DNA DAMAGE INDUCED CELL CYCLE G2 CHECKPOINT AND/OR AUGMENT ANTI-CANCER ACTIVITY OF DNA-DAMAGING TREATMENTS CDC25C, CHEK1, CDC25A HPGD 1650/4885KMT2A 883/4885SMN1; SMN2 4247/4885
US-20060122269-A1 Compounds that abrogate DNA damage induced cell cycle G2 checkpoint and/or augment anti-cancer activity of DNA-damaging treatments CDC25C, CHEK1, CDC25A HPGD 1650/4885KMT2A 883/4885SMN1; SMN2 4247/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.