SCHEMBL532820

SCHEMBL532820

COc1ccc(-c2nn3c(-c4cnc(NCCN(C)C)nc4)cnc3s2)cc1OC.COc1ccc(-c2nn3c(-c4cnc([S+](C)[O-])nc4)cnc3s2)cc1OC

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 6/20 0.51
FYN P06241 9/20 0.46
MKNK1 Q9BUB5 1/20 0.41
MKNK2 Q9HBH9 1/20 0.41
KDM4E B2RXH2 3/20 0.39
ALDH1A1 P00352 2/20 0.39
PKM P14618 1/20 0.39
HPGD P15428 1/20 0.39
STAT6 P42226 1/20 0.39
USP2 O75604 1/20 0.38
LMNA P02545 1/20 0.38
TSHR P16473 1/20 0.38
MAPK1 P28482 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
HSD17B10 Q99714 1/20 0.38
KMT2A Q03164 2/20 0.38
MEN1 O00255 1/20 0.38
DCTPP1 Q9H773 1/20 0.38
POLB P06746 1/20 0.37
RAD52 P43351 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2123416 0.92 PIK3CA (0.58) PIK3CAFYNMKNK1MKNK2KDM4E
SCHEMBL2120454 0.87 PIK3CA (0.64) PIK3CAFYNKDM4EALDH1A1PKM
SCHEMBL2123426 0.76 KDM4E (0.44) PIK3CAFYNMKNK1KDM4EALDH1A1
SCHEMBL532633 0.75 PIK3CA (0.74) PIK3CAFYNKDM4EALDH1A1PKM
SCHEMBL532289 0.71 PIK3CA (0.67) PIK3CAFYNKDM4EALDH1A1PKM
SCHEMBL2120460 0.69 KDM4E (0.49) PIK3CAKDM4EALDH1A1PKMHPGD
SCHEMBL532198 0.69 PIK3CA (0.61) PIK3CAFYNKDM4EALDH1A1PKM
SCHEMBL532016 0.68 PIK3CA (1.00) PIK3CAFYNKDM4EALDH1A1PKM
SCHEMBL533182 0.68 PIK3CA (0.71) PIK3CAFYNMKNK1MKNK2KDM4E
SCHEMBL15975809 0.68 PIK3CA (0.77) PIK3CAFYNMKNK1MKNK2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2414369-A1 IMIDAZO [2, 1-B][ 1, 3, 4]THIADIAZOLE DERIVATIVES Centro Nacional de Investigaciones Oncológicas (CNIO) (ES) 2012-02-08 EP disclosed
WO-2010112874-A1 IMIDAZO [2, 1-B] [ 1, 3, 4 ] THIADIAZOLE DERIVATIVES CENTRO NACIONAL DE INVESTIGACIONES ONCOLOGICAS (CNIO) (ES) 2010-10-07 WO disclosed