SCHEMBL5328631

SCHEMBL5328631

CN1Cc2cc(C(=O)O)ccc2NC1=O

nearest known ligand 0.62

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 18/20 0.62
CREBBP Q92793 2/20 0.54
BRD2 P25440 1/20 0.47
KDM4E B2RXH2 1/20 0.45
MAPT P10636 1/20 0.45
HPGD P15428 1/20 0.44
GFER P55789 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31490089 0.88 BRD4 (0.54) BRD4CREBBP
SCHEMBL7413152 0.84 BRD4 (0.54) BRD4CREBBPBRD2
SCHEMBL9768375 0.84 BRD4 (0.56) BRD4CREBBPBRD2MAPTHPGD
SCHEMBL7423824 0.84 BRD4 (0.60) BRD4CREBBPBRD2HPGDGFER
SCHEMBL7409687 0.81 BRD4 (0.57) BRD4CREBBPBRD2HPGDGFER
SCHEMBL4024924 0.81 KDM4E (0.49) BRD4KDM4EMAPT
SCHEMBL4024521 0.79 ITGB3 (0.47) BRD4
SCHEMBL10414690 0.78 BRD4 (0.50) BRD4CREBBP
SCHEMBL7434007 0.78 BRD4 (0.50) BRD4CREBBPBRD2
SCHEMBL7442306 0.78 BRD4 (0.50) BRD4CREBBPBRD2HPGDGFER

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007144379-A1 BICYCLIC COMPOUNDS USEFUL AS CATHEPSIN S INBHIBITORS MEDIVIR AB (SE) 2007-12-21 WO disclosed
WO-2007144379-A1 BICYCLIC COMPOUNDS USEFUL AS CATHEPSIN S INBHIBITORS MEDIVIR AB (SE) 2007-12-21 WO disclosed
WO-2006064286-A1 CATHEPSIN S INHIBITORS MEDIVIR UK LTD (GB) 2006-06-22 WO disclosed
WO-2006064286-A1 CATHEPSIN S INHIBITORS MEDIVIR UK LTD (GB) 2006-06-22 WO disclosed