SCHEMBL5330934

SCHEMBL5330934

O=C(CSc1nnc(-c2ccccc2)n1-c1cccnc1)N/N=C/c1ccco1

nearest known ligand 0.76

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.76
ALDH1A1 P00352 10/20 0.70
MAPT P10636 4/20 0.70
LMNA P02545 1/20 0.70
PTK2 Q05397 5/20 0.58
KMT2A Q03164 5/20 0.58
MEN1 O00255 4/20 0.58
HPGD P15428 1/20 0.58
POLB P06746 5/20 0.55
TDP1 Q9NUW8 4/20 0.55
SMN1; SMN2 Q16637 2/20 0.55
RECQL P46063 2/20 0.55
KDM4E B2RXH2 1/20 0.55
L3MBTL1 Q9Y468 1/20 0.55
HTT P42858 1/20 0.54
PKM P14618 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5330937 1.00 TP53 (0.76) TP53ALDH1A1MAPTLMNAPTK2
SCHEMBL14542267 0.87 TP53 (0.79) TP53ALDH1A1MAPTLMNAPTK2
SCHEMBL14542024 0.86 TP53 (0.78) TP53ALDH1A1MAPTLMNAPTK2
SCHEMBL5328282 0.84 TP53 (0.75) TP53ALDH1A1MAPTLMNAKMT2A
SCHEMBL5328274 0.84 TP53 (0.75) TP53ALDH1A1MAPTLMNAKMT2A
SCHEMBL13856360 0.81 PTK2 (0.77) ALDH1A1MAPTLMNAPTK2KMT2A
SCHEMBL5334648 0.81 MEN1 (0.81) TP53ALDH1A1MAPTPTK2KMT2A
SCHEMBL14542106 0.80 TP53 (0.69) TP53ALDH1A1MAPTLMNAPTK2
SCHEMBL14542264 0.80 HPGD (0.65) TP53ALDH1A1MAPTLMNAKMT2A
SCHEMBL14542416 0.80 TP53 (0.69) TP53ALDH1A1MAPTLMNAPTK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007047394-A2 THIOTRIAZOLYL DERIVATIVES EPIX DELAWARE, INC. (US) 2007-04-26 WO claimed
WO-2007047394-A2 THIOTRIAZOLYL DERIVATIVES EPIX DELAWARE, INC. (US) 2007-04-26 WO disclosed
WO-2007047394-A2 THIOTRIAZOLYL DERIVATIVES EPIX DELAWARE, INC. (US) 2007-04-26 WO disclosed