SCHEMBL5334758

SCHEMBL5334758

CC(C)(C)OC(=O)n1c(-c2cccc3c2C(=O)NC3)c(OCc2ccccc2)c2ccccc21

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 4/20 0.43
AURKA O14965 2/20 0.43
CCNB2 O95067 1/20 0.38
CDK1 P06493 1/20 0.38
CCNB1 P14635 1/20 0.38
GSK3B P49841 1/20 0.38
CCNB3 Q8WWL7 1/20 0.38
TRPV3 Q8NET8 1/20 0.36
CHRM2 P08172 1/20 0.36
CHRM4 P08173 1/20 0.36
CHRM1 P11229 1/20 0.36
CHRM3 P20309 1/20 0.36
USP2 O75604 1/20 0.35
ALDH1A1 P00352 1/20 0.35
TSHR P16473 1/20 0.35
HSD17B10 Q99714 1/20 0.35
ACHE P22303 1/20 0.35
NTRK1 P04629 1/20 0.35
GLP1R P43220 1/20 0.34
HDAC6 Q9UBN7 3/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5328430 0.77 AURKA (0.55) KDRAURKANR1H2GHSRBRD4
SCHEMBL5330620 0.73 BRD4 (0.55) NR1H2BRD4CREBBP
SCHEMBL5334220 0.70 AURKA (0.46) KDRAURKANR1H2GHSRBRD4
SCHEMBL3047240 0.70 CCNB2 (0.40) CCNB2CDK1CCNB1GSK3BCCNB3
SCHEMBL5327530 0.69 AURKA (0.48) KDRAURKACDK1NR1H2BRD4
SCHEMBL5331753 0.67 AURKA (0.42) KDRAURKACDK1PARP1MAPK1
SCHEMBL5331995 0.66 AURKA (0.42) KDRAURKANR1H2GHSRBRD4
SCHEMBL5333314 0.66 KDR (0.52) KDRAURKANR1H2BRD4CREBBP
SCHEMBL3840883 0.66 PARP1 (0.36) PARP1NR1H2BRD4CREBBP
SCHEMBL5334755 0.66 KDR (0.40) KDRAURKACDK1PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007047646-A2 SUBSTITUTED DIHYDRO-ISOINDOLONES USEFUL IN TREATING KINASE DISORDERS JANSSEN PHARMACEUTICA, N.V. (BE) 2007-04-26 WO disclosed