SCHEMBL5334755

SCHEMBL5334755

CC(C)(C)OC(=O)[N+]1(OCc2ccccc2)C(c2cccc3c2C(=O)NC3)=Cc2ccccc21

nearest known ligand 0.40

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KDR P35968 9/20 0.40
AURKA O14965 8/20 0.40
CDK1 P06493 1/20 0.33
CA12 O43570 1/20 0.32
CA9 Q16790 1/20 0.32
PARP1 P09874 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5328430 0.66 AURKA (0.55) KDRAURKA
SCHEMBL5334758 0.66 KDR (0.43) KDRAURKACDK1PARP1
SCHEMBL29029873 0.65 CA12 (0.60) KDRAURKACA12CA9PARP1
SCHEMBL5331753 0.62 AURKA (0.42) KDRAURKACDK1CA12CA9
SCHEMBL5330620 0.61 BRD4 (0.55) CA12CA9
SCHEMBL2980978 0.60 ALDH1A1 (0.39) CA12
SCHEMBL30775231 0.60 AURKA (0.61) KDRAURKACDK1CA12CA9
Bicarbonate SCHEMBL29928922 0.58 CA12 (0.84) KDRAURKACA12CA9PARP1
Bicarbonate SCHEMBL21081705 0.58 CA12 (0.84) KDRAURKACA12CA9PARP1
SCHEMBL8216557 0.57 ALDH1A1 (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007047646-A2 SUBSTITUTED DIHYDRO-ISOINDOLONES USEFUL IN TREATING KINASE DISORDERS JANSSEN PHARMACEUTICA, N.V. (BE) 2007-04-26 WO disclosed